SCHEMBL16843

SCHEMBL16843

C[C@H]1CN(C(=O)OC(C)(C)C)CCN1

nearest known ligand 0.50

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
NR1H2 P55055 1/20 0.47
USP2 O75604 1/20 0.46
SMN1; SMN2 Q16637 1/20 0.46
MAPK1 P28482 1/20 0.43
HPGD P15428 1/20 0.43
MAPT P10636 2/20 0.43
MEN1 O00255 1/20 0.43
ALDH1A1 P00352 1/20 0.43
KMT2A Q03164 1/20 0.43
RECQL P46063 1/20 0.41
EPHX1 P07099 1/20 0.41
BIRC2 Q13490 1/20 0.41
KDM4E B2RXH2 1/20 0.40
THRB P10828 1/20 0.40
EPHX2 P34913 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16018 1.00 NR1H2 (0.47) NR1H2USP2SMN1; SMN2MAPK1HPGD
SCHEMBL105348 1.00 NR1H2 (0.47) NR1H2USP2SMN1; SMN2MAPK1HPGD
Hydrochloric Acid SCHEMBL25337897 0.98 NR1H2 (0.46) NR1H2USP2SMN1; SMN2MAPK1HPGD
Piperazine SCHEMBL28853588 0.97 NR1H2 (0.45) NR1H2USP2SMN1; SMN2MAPK1HPGD
SCHEMBL28002373 0.97 HPGD (0.48) NR1H2USP2SMN1; SMN2MAPK1HPGD
Acetic Acid SCHEMBL28827133 0.95 NR1H2 (0.44) NR1H2USP2SMN1; SMN2MAPK1HPGD
Urea SCHEMBL4467391 0.95 NR1H2 (0.44) NR1H2USP2SMN1; SMN2MAPK1HPGD
Acetic Acid SCHEMBL28060582 0.95 NR1H2 (0.44) NR1H2USP2SMN1; SMN2MAPK1HPGD
SCHEMBL31540 0.90 HPGD (0.48) NR1H2USP2SMN1; SMN2MAPK1HPGD
SCHEMBL2898103 0.90 HPGD (0.48) NR1H2USP2SMN1; SMN2MAPK1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1952 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4234546-B1 IMPROVED SYNTHESIS OF KEY INTERMEDIATE OF KRAS G12C INHIBITOR COMPOUND AMGEN INC (US) 2026-04-15 EP claimed
US-20250388579-A1 SYNTHESIS OF KRAS G12C INHIBITOR COMPOUND AMGEN INC. (US) 2025-12-25 US claimed
US-20250368643-A1 SYNTHESIS OF KEY INTERMEDIATE OF KRAS G12C INHIBITOR COMPOUND AMGEN INC. (US) 2025-12-04 US claimed
US-12473281-B2 Synthesis of KRAS G12C inhibitor compound AMGEN INC. (US) 2025-11-18 US claimed
US-20250206736-A1 SYNTHESIS OF KRAS G12C INHIBITOR COMPOUND AMGEN INC. (US) 2025-06-26 US claimed
US-20250206735-A1 SYNTHESIS OF KEY INTERMEDIATE OF KRAS G12C INHIBITOR COMPOUND AMGEN INC. (US) 2025-06-26 US claimed
EP-4476205-A1 PROCESS FOR SYNTHESIS OF QUINAZOLINE COMPOUNDS Genentech Inc. (US) 2024-12-18 EP claimed
CN-118574820-A Method for synthesizing quinazoline compounds 基因泰克公司 2024-08-30 CN claimed
US-12071422-B2 Process for synthesis of quinazoline compounds GENENTECH, INC. (US) 2024-08-27 US claimed
CN-117903117-A Preparation method of KRAS G12C inhibitor divarasib 云南万宏医药科技有限公司 2024-04-19 CN claimed
CN-115466259-B Preparation method of KRAS G12C inhibitor sotorubin 山东大学 2023-12-05 CN claimed
EP-4234546-A2 IMPROVED SYNTHESIS OF KEY INTERMEDIATE OF KRAS G12C INHIBITOR COMPOUND Amgen Inc. (US) 2023-08-30 EP claimed
WO-2023150653-A1 PROCESS FOR SYNTHESIS OF QUINAZOLINE COMPOUNDS GENENTECH, INC. (US) 2023-08-10 WO claimed
US-20230250074-A1 PROCESS FOR SYNTHESIS OF QUINAZOLINE COMPOUNDS GENENTECH, INC. (US) 2023-08-10 US claimed
CN-115466259-A Preparation method of KRAS G12C inhibitor sotoxib 山东大学 2022-12-13 CN claimed
CN-114907387-A Pyrimidopyrrole KRAS inhibitor and preparation method and application thereof 中山大学 2022-08-16 CN claimed
CN-114057654-A Preparation method of (S) -1-Boc-3-methylpiperazine 苏州艾缇克药物化学有限公司 2022-02-18 CN claimed
CN-113754579-A Preparation method of pyridine derivative 正大天晴药业集团股份有限公司 2021-12-07 CN claimed
EP-4747245-A1 PHARMACEUTICAL COMPOUNDS Almac Discovery Limited (GB) 2026-05-27 EP disclosed
US-5712267-A Carbapenem derivatives, their preparation and their use as antibiotics SANKYO COMPANY,. LIMITED (JP) 1998-01-27 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (7 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-12071422-B2 Process for synthesis of quinazoline compounds HCCS, NQO2, SQLE NR1H2 2492/4885USP2 2729/4885SMN1; SMN2 3950/4885
US-20250368643-A1 SYNTHESIS OF KEY INTERMEDIATE OF KRAS G12C INHIBITOR COMPOUND KRAS, NRAS, HRAS NR1H2 4045/4885USP2 2323/4885SMN1; SMN2 3898/4885
US-20230250074-A1 PROCESS FOR SYNTHESIS OF QUINAZOLINE COMPOUNDS HCCS, NQO2, SQLE NR1H2 2492/4885USP2 2729/4885SMN1; SMN2 3950/4885
US-12473281-B2 Synthesis of KRAS G12C inhibitor compound KRAS, NRAS, HRAS NR1H2 3929/4885USP2 2447/4885SMN1; SMN2 2239/4885
US-20250206736-A1 SYNTHESIS OF KRAS G12C INHIBITOR COMPOUND KRAS, NRAS, HRAS NR1H2 3929/4885USP2 2447/4885SMN1; SMN2 2239/4885
US-20250206735-A1 SYNTHESIS OF KEY INTERMEDIATE OF KRAS G12C INHIBITOR COMPOUND KRAS, NRAS, HRAS NR1H2 4045/4885USP2 2323/4885SMN1; SMN2 3898/4885
US-20250388579-A1 SYNTHESIS OF KRAS G12C INHIBITOR COMPOUND KRAS, NRAS, BRAF NR1H2 2503/4885USP2 1581/4885SMN1; SMN2 3026/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.