SCHEMBL16856437

SCHEMBL16856437

O=C(O)C[C@H]1CNc2cc(I)ccc2O1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSD17B10 Q99714 1/20 0.37
HPGD P15428 3/20 0.35
CYP1A2 P05177 2/20 0.35
CYP2C9 P11712 2/20 0.35
CYP2C19 P33261 2/20 0.35
CYP3A4 P08684 1/20 0.35
KMT2A Q03164 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.34
DRD2 P14416 2/20 0.34
DRD1 P21728 2/20 0.34
DRD4 P21917 2/20 0.34
DRD5 P21918 2/20 0.34
DRD3 P35462 2/20 0.34
ITGB3 P05106 2/20 0.33
ITGA2B P08514 2/20 0.33
CYP2D6 P10635 1/20 0.33
AKR1B1 P15121 1/20 0.33
ADAMTS5 Q9UNA0 1/20 0.32
ALDH1A1 P00352 1/20 0.32
HTT P42858 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16856434 0.85 HPGD (0.36) HSD17B10HPGDCYP1A2CYP2C9CYP2C19
SCHEMBL16851256 0.84 USP2 (0.44) HSD17B10HPGDCYP1A2CYP2C9CYP2C19
SCHEMBL16851189 0.80 HSD17B10 (0.34) HSD17B10HPGDCYP1A2CYP2C9CYP2C19
SCHEMBL6860121 0.79 AKR1B1 (0.43) CYP1A2KMT2AAKR1B1ALDH1A1
Hydrochloric Acid SCHEMBL9153498 0.78 HPGD (0.48) HSD17B10HPGDSMN1; SMN2ALDH1A1HTT
SCHEMBL6860296 0.75 RORC (0.39) HSD17B10KMT2AITGB3ITGA2BRORC
SCHEMBL25072496 0.73 MIF (0.33) HPGDCYP1A2CYP2C9CYP2C19CYP2D6
SCHEMBL16851484 0.73 RORC (0.56) RORC
SCHEMBL90825 0.72 AR (0.51) HSD17B10CYP3A4DRD2DRD1DRD4
SCHEMBL34474543 0.70 TDP1 (0.41) HSD17B10HPGDCYP1A2CYP2C9CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015095792-A1 CARBAMATE BENZOXAXINE PROPIONIC ACIDS AND ACID DERIVATIVES FOR MODULATION OF RORGAMMA ACTIVITY AND THE TREATMENT OF DISEASE MERCK SHARP & DOHME CORP. (US) 2015-06-25 WO disclosed