SCHEMBL16857774

SCHEMBL16857774

O=C(O)Oc1cnn(-c2nc3ccc(OC4CCCCC4)cc3c(=O)[nH]2)c1

nearest known ligand 0.52

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
SPR P35270 2/20 0.52
EGLN1 Q9GZT9 16/20 0.49
KDM4C Q9H3R0 1/20 0.38
MAOB P27338 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3032298 0.88 EGLN1 (0.64) EGLN1
SCHEMBL16857823 0.86 EGLN1 (0.47) SPREGLN1
SCHEMBL16857699 0.83 EGLN1 (0.56) EGLN1
SCHEMBL16857824 0.82 EGLN1 (0.44) SPREGLN1
SCHEMBL16857877 0.82 EGLN1 (0.47) SPREGLN1
SCHEMBL16857775 0.81 EGLN1 (0.49) EGLN1KDM4C
SCHEMBL16857869 0.81 EGLN1 (0.47) EGLN1
SCHEMBL16857708 0.81 MGLL (0.45) EGLN1
SCHEMBL16857875 0.81 EGLN1 (0.47) EGLN1
SCHEMBL16857832 0.81 EGLN1 (0.58) EGLN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2396316-B1 QUINAZOLINONES AS PROLYL HYDROXYLASE INHIBITORS JANSSEN PHARMACEUTICA NV (BE) 2015-07-01 EP claimed