SCHEMBL16858397

SCHEMBL16858397

COc1ccc2c(c1)C(=O)N(CC1CCCCC1)C2

nearest known ligand 0.54

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
ADAM17 P78536 14/20 0.54
OPRM1 P35372 3/20 0.46
OPRL1 P41146 2/20 0.46
OPRK1 P41145 1/20 0.46
TNF P01375 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL5252190 0.86 ADAM17 (0.52) ADAM17TNF
SCHEMBL16820515 0.84 ADAM17 (0.47) ADAM17TNF
SCHEMBL16820518 0.84 ADAM17 (0.47) ADAM17TNF
SCHEMBL16858382 0.83 ADAM17 (0.47) ADAM17
SCHEMBL16820419 0.83 ADAM17 (0.47) ADAM17TNF
SCHEMBL16820418 0.83 ADAM17 (0.47) ADAM17TNF
SCHEMBL16850270 0.80 CRBN (0.44) ADAM17OPRM1OPRL1OPRK1
SCHEMBL16820474 0.80 ADAM17 (0.44) ADAM17TNF
SCHEMBL16820473 0.80 ADAM17 (0.44) ADAM17TNF
SCHEMBL16850271 0.80 CRBN (0.44) ADAM17OPRM1OPRL1OPRK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015095052-A1 ISOINDOLIN-1-ONES AS MACROPHAGE MIGRATION INHIBITORY FACTOR (MIF) INHIBITORS CONTROLLED CHEMICALS, INC. (US) 2015-06-25 WO disclosed