SCHEMBL1687286

SCHEMBL1687286

CN(c1cccc(CS(C)(=O)=O)c1)c1nc(N)ncc1-c1ccc2cn[nH]c2c1

nearest known ligand 0.39

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
FGFR1 P11362 4/20 0.39
FGFR2 P21802 2/20 0.39
USP7 Q93009 2/20 0.39
PIK3CD O00329 3/20 0.39
PIK3CB P42338 3/20 0.39
PIK3CA P42336 2/20 0.39
PIK3CG P48736 2/20 0.39
MKNK1 Q9BUB5 2/20 0.38
MKNK2 Q9HBH9 2/20 0.38
FGFR3 P22607 1/20 0.38
LCK P06239 1/20 0.37
BTK Q06187 1/20 0.37
CDK2 P24941 1/20 0.35
CLK1 P49759 1/20 0.35
DYRK1A Q13627 1/20 0.35
CLK4 Q9HAZ1 1/20 0.35
DDR2 Q16832 1/20 0.35
MAPKAPK2 P49137 2/20 0.35
CSF1R P07333 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29430391 0.72 PIK3CD (0.51) FGFR1FGFR2USP7PIK3CDPIK3CB
SCHEMBL4476790 0.72 PIK3CD (0.51) FGFR1FGFR2USP7PIK3CDPIK3CB
SCHEMBL588382 0.71 PKMYT1 (0.49) FGFR1FGFR2PIK3CDPIK3CBPIK3CA
SCHEMBL31672542 0.69 KDR (0.64)
SCHEMBL10151186 0.69 KDR (0.64)
SCHEMBL2745386 0.68 DHFR (0.59) FGFR1FGFR2USP7PIK3CDPIK3CB
Hydrochloric Acid SCHEMBL4478858 0.67 DHFR (0.57) FGFR1FGFR2USP7PIK3CDPIK3CB
Hydrochloric Acid SCHEMBL29430410 0.67 DHFR (0.57) FGFR1FGFR2USP7PIK3CDPIK3CB
Hydrochloric Acid SCHEMBL4478855 0.66 DHFR (0.56) FGFR1FGFR2USP7PIK3CDPIK3CB
SCHEMBL6810597 0.63 KDR (0.41) FGFR1FGFR2FGFR3LCKDDR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2311825-A1 Pyrimidineamines as angiogenesis modulators GlaxoSmithKline LLC (US) 2011-04-20 EP claimed