SCHEMBL1688159

SCHEMBL1688159

CN1CC2(CCN(Cc3ccc(CN)cc3)CC2)c2ccccc21

nearest known ligand 0.66

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 3/20 0.66
HDAC6 Q9UBN7 3/20 0.66
HDAC8 Q9BY41 1/20 0.66
SIGMAR1 Q99720 11/20 0.54
SLC18A3 Q16572 7/20 0.54
FFAR1 O14842 1/20 0.49
OPRL1 P41146 1/20 0.46
ALDH1A1 P00352 1/20 0.46
TP53 P04637 1/20 0.46
CYP1A2 P05177 1/20 0.46
CYP3A4 P08684 1/20 0.46
CYP2D6 P10635 1/20 0.46
CYP2C9 P11712 1/20 0.46
TSHR P16473 1/20 0.46
CYP2C19 P33261 1/20 0.46
CA2 P00918 1/20 0.46
NCF1 P14598 1/20 0.46
CHKA P35790 1/20 0.46
PRMT6 Q96LA8 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1980590 0.89 HDAC1 (0.68) HDAC1HDAC6HDAC8SIGMAR1SLC18A3
SCHEMBL13519235 0.87 HDAC1 (0.69) HDAC1HDAC6HDAC8SIGMAR1SLC18A3
SCHEMBL15494623 0.85 HDAC1 (0.64) HDAC1HDAC6HDAC8SIGMAR1SLC18A3
SCHEMBL15160327 0.85 HDAC1 (0.67) HDAC1HDAC6HDAC8SIGMAR1SLC18A3
SCHEMBL17117621 0.83 HDAC1 (0.64) HDAC1HDAC6HDAC8SIGMAR1SLC18A3
SCHEMBL13518796 0.83 HDAC1 (0.78) HDAC1HDAC6HDAC8SIGMAR1SLC18A3
SCHEMBL15158679 0.82 HDAC1 (0.63) HDAC1HDAC6HDAC8SIGMAR1SLC18A3
SCHEMBL11472209 0.77 SIGMAR1 (0.68) HDAC1HDAC6HDAC8SIGMAR1SLC18A3
SCHEMBL13519118 0.77 HDAC1 (0.57) HDAC1HDAC6HDAC8SIGMAR1SLC18A3
SCHEMBL12716195 0.76 SIGMAR1 (0.59) HDAC1HDAC6HDAC8SIGMAR1SLC18A3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012046869-A1 CYCLIC AMIDE DERIVATIVE 持田製薬株式会社 (JP) 2012-04-12 WO disclosed