SCHEMBL16888498

SCHEMBL16888498

C=C(C)c1cnc(-c2cc(Cl)ccc2F)cc1Nc1ncnc2c1CN2

nearest known ligand 0.56

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
TGFBR1 P36897 20/20 0.56
ACVR1B P36896 14/20 0.56
ACVRL1 P37023 10/20 0.56
ACVR1 Q04771 3/20 0.56
CYP3A4 P08684 1/20 0.40
CYP2C8 P10632 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16879277 0.81 TGFBR1 (0.56) TGFBR1ACVR1BACVRL1ACVR1CYP3A4
SCHEMBL16879809 0.81 TGFBR1 (0.56) TGFBR1ACVR1BACVRL1ACVR1
SCHEMBL16879186 0.77 TGFBR1 (0.72) TGFBR1ACVR1BACVRL1ACVR1
SCHEMBL16879709 0.76 TGFBR1 (0.56) TGFBR1ACVR1BACVRL1ACVR1
SCHEMBL18219801 0.75 TGFBR1 (0.68) TGFBR1ACVR1BACVRL1ACVR1CYP3A4
SCHEMBL16879552 0.75 TGFBR1 (0.57) TGFBR1ACVR1BACVRL1ACVR1
SCHEMBL16879826 0.74 TGFBR1 (0.59) TGFBR1ACVR1BACVRL1ACVR1CYP3A4
SCHEMBL16879672 0.74 TGFBR1 (0.66) TGFBR1ACVR1BACVRL1ACVR1CYP3A4
SCHEMBL16879389 0.74 TGFBR1 (0.54) TGFBR1ACVR1BACVRL1ACVR1CYP3A4
SCHEMBL20397408 0.74 TGFBR1 (0.59) TGFBR1ACVR1BACVRL1ACVR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015103355-A1 COMPOUNDS AND METHODS OF USE MEDIVATION TECHNOLOGIES, INC. (US) 2015-07-09 WO disclosed