SCHEMBL16893103

SCHEMBL16893103

Cc1cccc(-c2cnc(N)nc2-c2c[nH]c(OC(=O)N(C)Cc3ccccc3)c2)c1

nearest known ligand 0.54

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
ADORA1 P30542 12/20 0.54
ADORA2A P29274 8/20 0.42
MAPT P10636 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39
ABHD6 Q9BV23 1/20 0.39
MAPK1 P28482 1/20 0.39
LMNA P02545 1/20 0.38
GAA P10253 1/20 0.38
MAPK10 P53779 1/20 0.38
CNR1 P21554 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16893064 0.93 MAPT (0.45) ADORA1ADORA2AMAPTNPSR1ABHD6
SCHEMBL16893040 0.91 ADORA1 (0.53) ADORA1ADORA2AMAPTNPSR1MAPK1
SCHEMBL16893046 0.86 ADORA1 (0.56) ADORA1ADORA2AMAPTNPSR1GAA
SCHEMBL5412959 0.86 ADORA1 (0.56) ADORA1ADORA2AMAPK1CNR1
SCHEMBL16893097 0.84 MAPK1 (0.37) ADORA1ADORA2AMAPTNPSR1ABHD6
SCHEMBL16893055 0.81 ADORA1 (0.49) ADORA1ADORA2AMAPTNPSR1LMNA
SCHEMBL5400627 0.78 MAPK1 (0.54) ADORA1ADORA2AMAPTNPSR1MAPK1
SCHEMBL16893005 0.77 ABHD6 (0.42) ADORA2AABHD6
SCHEMBL5412969 0.77 MAPK1 (0.67) ADORA1ADORA2AMAPK1MAPK10
SCHEMBL5397397 0.76 ADORA1 (0.66) ADORA1ADORA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1363906-B1 HETEROCYCLIC INHIBITORS OF ERK2 AND USES THEREOF VERTEX PHARMA (US) 2015-07-15 EP claimed