SCHEMBL1689458

SCHEMBL1689458

NC(=O)C(C(=O)Nc1nc(-c2ccccc2)cs1)(c1ccc(C(=O)Nc2ccccc2N)cc1)c1nc(-c2ccccc2)cs1

nearest known ligand 0.61

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
HDAC3 O15379 1/20 0.61
HDAC1 Q13547 1/20 0.61
HDAC2 Q92769 1/20 0.61
HDAC8 Q9BY41 1/20 0.61
SCD O00767 1/20 0.52
PARP1 P09874 1/20 0.49
PHGDH O43175 3/20 0.48
ADORA3 P0DMS8 1/20 0.48
RAB9A P51151 2/20 0.46
MAPT P10636 2/20 0.46
KDM4E B2RXH2 1/20 0.46
NPC1 O15118 1/20 0.46
PKM P14618 1/20 0.46
SMN1; SMN2 Q16637 1/20 0.46
MEN1 O00255 2/20 0.45
KMT2A Q03164 2/20 0.45
GAA P10253 1/20 0.45
LMNA P02545 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2108677 0.77 HDAC1 (0.67) HDAC3HDAC1HDAC2HDAC8SCD
SCHEMBL16892942 0.73 ALDH1A1 (0.51) ADORA3RAB9AMAPTKDM4ENPC1
SCHEMBL23674562 0.72 SCD (0.84) SCDPARP1PHGDHADORA3RAB9A
SCHEMBL1270375 0.71 SCD (0.89) SCDPARP1PHGDHADORA3RAB9A
SCHEMBL31265595 0.71 PARP1 (0.74) SCDPARP1PHGDHADORA3RAB9A
SCHEMBL233522 0.71 SCD (0.78) SCDPARP1PHGDHADORA3RAB9A
SCHEMBL13206963 0.71 SCD (0.82) SCDPARP1PHGDHADORA3RAB9A
SCHEMBL8349704 0.70 HDAC1 (0.87) HDAC3HDAC1HDAC2HDAC8RAB9A
SCHEMBL16562127 0.70 SCD (1.00) SCDPARP1PHGDHADORA3RAB9A
SCHEMBL1065242 0.69 HDAC1 (0.85) HDAC3HDAC1HDAC2HDAC8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1896395-A2 MODIFIED MALONATE DERIVATIVES Merck & Co., Inc. (US) 2008-03-12 EP claimed
WO-2007002248-A2 MODIFIED MALONATE DERIVATIVES MERCK & CO., INC. (US) 2007-01-04 WO claimed