SCHEMBL16908014

SCHEMBL16908014

NC(=O)C[C@H](NC(=O)C(F)(F)F)C(N)=O

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ECE1 P42892 3/20 0.42
ITGB2 P05107 2/20 0.35
ICAM1 P05362 2/20 0.35
ITGAL P20701 2/20 0.35
CA2 P00918 4/20 0.34
ALDH1A1 P00352 2/20 0.34
POLB P06746 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33
GRB2 P62993 1/20 0.33
SCN9A Q15858 2/20 0.33
ESR1 P03372 1/20 0.32
KCNH2 Q12809 1/20 0.32
CA3 P07451 2/20 0.31
CA5A P35218 2/20 0.31
CA5B Q9Y2D0 2/20 0.31
CA12 O43570 1/20 0.31
CA4 P22748 1/20 0.31
CA6 P23280 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6620751 0.86 ITGB2 (0.47) ECE1ITGB2ICAM1ITGALCA2
SCHEMBL6620753 0.86 ITGB2 (0.47) ECE1ITGB2ICAM1ITGALCA2
SCHEMBL19463542 0.86 ITGB2 (0.47) ECE1ITGB2ICAM1ITGALCA2
SCHEMBL11401620 0.83 ITGB2 (0.33) ECE1ITGB2ICAM1ITGALCA2
SCHEMBL5777336 0.83 ECE1 (0.44) ECE1ITGB2ICAM1ITGALCA2
SCHEMBL6623611 0.82 FOLH1 (0.35) ECE1ITGB2ICAM1ITGALCA2
SCHEMBL6623613 0.82 FOLH1 (0.35) ECE1ITGB2ICAM1ITGALCA2
SCHEMBL17697188 0.81 PTPN1 (0.37) CA2ALDH1A1POLBSMN1; SMN2MEN1
SCHEMBL10993372 0.80 SMN1; SMN2 (0.35) CA2ALDH1A1POLBSMN1; SMN2MEN1
SCHEMBL7349775 0.80 ECE1 (0.46) ECE1ITGB2ICAM1ITGALCA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015106200-A2 DIPEPTIDES AS INHIBITORS OF HUMAN IMMUNOPROTEASOMES CORNELL UNIVERSITY (US) 2015-07-16 WO disclosed