SCHEMBL169122

SCHEMBL169122

O=C(O)CN1CCOC(CO)C1

nearest known ligand 0.48

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
HSD17B10 Q99714 1/20 0.48
PDK1 Q15118 2/20 0.45
HRH3 Q9Y5N1 1/20 0.41
DRD4 P21917 2/20 0.36
ADORA2A P29274 2/20 0.35
ADORA1 P30542 2/20 0.35
ADORA3 P0DMS8 1/20 0.35
ADORA2B P29275 1/20 0.35
GLA P06280 1/20 0.34
DRD2 P14416 1/20 0.34
DRD3 P35462 1/20 0.34
HDAC6 Q9UBN7 1/20 0.34
KDM4E B2RXH2 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28864592 1.00 HSD17B10 (0.48) HSD17B10PDK1HRH3DRD4ADORA2A
SCHEMBL12226473 0.84 PDK1 (0.44) PDK1HRH3DRD4ADORA2AADORA1
SCHEMBL6966556 0.84 HSD17B10 (0.47) HSD17B10PDK1DRD4GLADRD2
SCHEMBL12226471 0.84 PDK1 (0.44) PDK1HRH3DRD4ADORA2AADORA1
SCHEMBL12226474 0.84 PDK1 (0.44) PDK1HRH3DRD4ADORA2AADORA1
SCHEMBL23299347 0.81 HSD17B10 (0.44) HSD17B10PDK1DRD4DRD2DRD3
SCHEMBL27687249 0.80 PDK1 (0.46) PDK1HRH3DRD4ADORA2AADORA1
SCHEMBL28153145 0.80 PDK1 (0.46) PDK1HRH3DRD4ADORA2AADORA1
SCHEMBL27687247 0.80 PDK1 (0.46) PDK1HRH3DRD4ADORA2AADORA1
SCHEMBL9281464 0.79 HSD17B10 (0.54) HSD17B10DRD4GLADRD2DRD3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102656179-A Bufalin derivatives, pharmaceutical compositions and uses thereof SUZHOU NEUPHARMA CO LTD 2012-09-05 CN claimed
WO-2012027957-A1 BUFALIN DERIVATIVES, PHARMACEUTICAL COMPOSITIONS AND USE THEREOF SUZHOU NEUPHARMA CO., LTD. (CN) 2012-03-08 WO claimed
CN-102656179-B Bufalin derivatives, pharmaceutical compositions and uses thereof SUZHOU NEUPHARMA Co.,Ltd. (CN) 2015-07-29 CN disclosed
CN-102656179-A Bufalin derivatives, pharmaceutical compositions and uses thereof SUZHOU NEUPHARMA CO LTD 2012-09-05 CN disclosed