SCHEMBL1692123

SCHEMBL1692123

CC(C)OCC1(C(=O)c2ccc3c(cnn3[Si](C(C)C)(C(C)C)C(C)C)c2)CCCN1C(=O)O

nearest known ligand 0.33

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 1/20 0.33
SLC6A2 P23975 1/20 0.33
SLC6A4 P31645 1/20 0.33
SLC6A3 Q01959 1/20 0.33
KDM2B Q8NHM5 3/20 0.32
TNKS O95271 1/20 0.31
TNKS2 Q9H2K2 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL443130 0.90 GPR119 (0.31) CYP2D6SLC6A2SLC6A4SLC6A3KDM2B
SCHEMBL443798 0.78 CNR2 (0.36) KDM2B
SCHEMBL440868 0.78 CNR2 (0.34) KDM2B
SCHEMBL445011 0.72 GPR119 (0.33)
SCHEMBL442649 0.69 CYP2D6 (0.47) CYP2D6SLC6A2SLC6A4SLC6A3
SCHEMBL446236 0.66 GPR119 (0.33)
SCHEMBL444471 0.65
SCHEMBL443784 0.64 CNR2 (0.35)
SCHEMBL24339380 0.60 SLC22A12 (0.43)
SCHEMBL1692041 0.59 CNR2 (0.34) CYP2D6SLC6A2SLC6A4SLC6A3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2297096-A2 ARYL KETONE AS MRI F. Hoffmann-La Roche AG (CH) 2011-03-23 EP disclosed
WO-2009153178-A2 ARYL KETONE AS MRI F. HOFFMANN-LA ROCHE AG (CH) 2009-12-23 WO disclosed