SCHEMBL16936786

SCHEMBL16936786

CC(C)(C)N1CCC(O)(c2ccc(Cl)cc2)C1

nearest known ligand 0.51

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
MAPT P10636 2/20 0.51
CCR3 P51677 1/20 0.50
OPRL1 P41146 5/20 0.49
OPRM1 P35372 3/20 0.49
OPRD1 P41143 1/20 0.49
OPRK1 P41145 1/20 0.49
DRD2 P14416 4/20 0.49
SLC18A3 Q16572 1/20 0.48
KMT2A Q03164 3/20 0.46
MEN1 O00255 2/20 0.46
ALDH1A1 P00352 1/20 0.45
LMNA P02545 1/20 0.45
POLB P06746 1/20 0.45
TSHR P16473 1/20 0.45
HTT P42858 1/20 0.45
HSD17B10 Q99714 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15543779 0.92 MAPT (0.55) MAPTCCR3OPRL1OPRM1OPRD1
SCHEMBL24422207 0.83 OPRM1 (0.59) OPRL1OPRM1OPRD1OPRK1ALDH1A1
SCHEMBL9910960 0.78 CCR3 (0.50) MAPTCCR3OPRL1OPRM1OPRD1
SCHEMBL3591425 0.78 CCR3 (0.57) CCR3OPRL1OPRM1OPRD1OPRK1
SCHEMBL18026610 0.76 CCR3 (0.60) CCR3OPRL1OPRM1DRD2
SCHEMBL8026713 0.76 OPRM1 (0.54) MAPTOPRL1OPRM1OPRD1OPRK1
SCHEMBL24421698 0.76 OPRM1 (0.49) MAPTOPRL1OPRM1OPRD1OPRK1
SCHEMBL17886542 0.75 OPRM1 (0.46) OPRL1OPRM1OPRD1OPRK1
SCHEMBL19462825 0.75 OPRM1 (0.43) OPRL1OPRM1OPRD1OPRK1DRD2
SCHEMBL16936710 0.75 OPRM1 (0.53) OPRL1OPRM1OPRD1OPRK1DRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3096754-A1 METALLO-BETA-LACTAMASE INHIBITORS Merck Sharp & Dohme Corp. (US) 2016-11-30 EP disclosed
WO-2015112441-A1 METALLO-BETA-LACTAMASE INHIBITORS MERCK SHARP & DOHME CORP. (US) 2015-07-30 WO disclosed