SCHEMBL169396

SCHEMBL169396

CCc1nc2c(N3CCOCC3)nc(SCc3ccc(OC)cc3)nc2n1CCN

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.49
NPSR1 Q6W5P4 3/20 0.49
PDE10A Q9Y233 2/20 0.43
TSHR P16473 3/20 0.40
HPGD P15428 2/20 0.40
HSD17B10 Q99714 2/20 0.40
PIK3CA P42336 2/20 0.39
NOS1 P29475 1/20 0.39
HDAC1 Q13547 4/20 0.39
LMNA P02545 2/20 0.39
HTT P42858 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
PIK3CD O00329 1/20 0.38
PIK3R1 P27986 1/20 0.38
NPC1 O15118 1/20 0.37
RAB9A P51151 1/20 0.37
HDAC3 O15379 1/20 0.37
HDAC4 P56524 1/20 0.37
HDAC7 Q8WUI4 1/20 0.37
HDAC2 Q92769 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL98830 0.93 ALDH1A1 (0.49) ALDH1A1NPSR1PDE10ATSHRHPGD
SCHEMBL98561 0.93 ALDH1A1 (0.50) ALDH1A1NPSR1PDE10ATSHRHPGD
SCHEMBL98635 0.88 ALDH1A1 (0.52) ALDH1A1NPSR1PDE10ATSHRHPGD
SCHEMBL98678 0.86 ALDH1A1 (0.44) ALDH1A1NPSR1PDE10ATSHRHPGD
SCHEMBL98260 0.84 ALDH1A1 (0.50) ALDH1A1NPSR1PDE10ATSHRHPGD
SCHEMBL97423 0.83 ALDH1A1 (0.51) ALDH1A1NPSR1PDE10ATSHRHPGD
SCHEMBL98691 0.83 PDE10A (0.55) ALDH1A1NPSR1PDE10ATSHRHPGD
SCHEMBL98831 0.82 PDE10A (0.41) ALDH1A1PDE10ATSHRHPGDHSD17B10
SCHEMBL98731 0.81 ALDH1A1 (0.47) ALDH1A1NPSR1PDE10ATSHRHPGD
SCHEMBL99966 0.81 ALDH1A1 (0.54) ALDH1A1NPSR1PDE10ATSHRHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2426130-A1 PURINE DERIVATIVE AND ANTITUMOR AGENT USING SAME ZENYAKU KOGYO KABUSHIKIKAISHA (JP) 2012-03-07 EP disclosed