SCHEMBL1695997

SCHEMBL1695997

COC(=O)c1sccc1N(CC(=O)O[C@H]1CN2CCC1CC2)c1ccc(OC)nc1

nearest known ligand 0.39

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
CHRM2 P08172 8/20 0.39
CHRM1 P11229 8/20 0.39
CHRM3 P20309 8/20 0.39
CHRM5 P08912 2/20 0.39
CHRM4 P08173 1/20 0.39
CYP2D6 P10635 1/20 0.39
NTMT1 Q9BV86 1/20 0.37
RAB9A P51151 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1696114 1.00 CHRM2 (0.39) CHRM2CHRM1CHRM3CHRM5CHRM4
SCHEMBL1696221 0.86 CYP2D6 (0.43) CHRM2CHRM1CHRM3CHRM5CHRM4
SCHEMBL1696085 0.85 CHRM2 (0.51) CHRM2CHRM1CHRM3CHRM5CHRM4
SCHEMBL1696230 0.77 TSHR (0.42) CHRM2CHRM1CHRM3CHRM5CHRM4
SCHEMBL1696246 0.77 TSHR (0.42) CHRM2CHRM1CHRM3CHRM5CHRM4
SCHEMBL16461576 0.73 NTMT1 (0.39) CHRM3NTMT1RAB9A
SCHEMBL1695999 0.73 NTMT1 (0.39) CHRM3NTMT1RAB9A
SCHEMBL1696267 0.73 NTMT1 (0.39) CHRM3NTMT1RAB9A
SCHEMBL2486589 0.67 CHRM2 (0.66) CHRM2CHRM1CHRM3CHRM5CHRM4
SCHEMBL2487397 0.64 CHRM2 (0.58) CHRM2CHRM1CHRM3CHRM5CHRM4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2585458-A1 ALKALOID AMINOESTER DERIVATIVES AND MEDICINAL COMPOSITION THEREOF Chiesi Farmaceutici S.p.A. (IT) 2013-05-01 EP disclosed
EP-2585457-A1 ALKALOID AMINOESTER DERIVATIVES AND MEDICINAL COMPOSITION THEREOF Chiesi Farmaceutici S.p.A. (IT) 2013-05-01 EP disclosed
WO-2011160918-A1 ALKALOID AMINOESTER DERIVATIVES AND MEDICINAL COMPOSITION THEREOF CHIESI FARMACEUTICI S.P.A. (IT) 2011-12-29 WO disclosed
WO-2011160919-A1 ALKALOID AMINOESTER DERIVATIVES AND MEDICINAL COMPOSITION THEREOF CHIESI FARMACEUTICI S.P.A. (IT) 2011-12-29 WO disclosed