SCHEMBL16972785

SCHEMBL16972785

Cc1c(Cl)cnc(Cl)c1Cl

nearest known ligand 0.48

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
PLAU P00749 1/20 0.48
DAO P14920 1/20 0.39
POLB P06746 2/20 0.33
MEN1 O00255 1/20 0.33
CYP1A2 P05177 1/20 0.33
CYP2C9 P11712 1/20 0.33
CYP2C19 P33261 1/20 0.33
KMT2A Q03164 1/20 0.33
L3MBTL1 Q9Y468 3/20 0.32
HPGD P15428 1/20 0.31
MAPK1 P28482 1/20 0.31
HTT P42858 1/20 0.31
BCL2L1 Q07817 1/20 0.30
MCL1 Q07820 1/20 0.30
ALDH1A1 P00352 1/20 0.30
MAPT P10636 1/20 0.30
NPSR1 Q6W5P4 1/20 0.30
DRD1 P21728 1/20 0.30
TDP1 Q9NUW8 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30039332 0.79 CCR1 (0.41) PLAUALDH1A1
SCHEMBL12139492 0.79 PLAU (0.48) PLAUDAOPOLBMEN1CYP1A2
SCHEMBL22129513 0.79 CCR1 (0.41) PLAUALDH1A1
SCHEMBL6664399 0.79 PLAU (0.44) PLAUDAOPOLBALDH1A1MAPT
SCHEMBL24844536 0.75 UHRF1 (0.38) PLAUALDH1A1TDP1
SCHEMBL31410007 0.75 DAO (0.37) PLAUDAOALDH1A1
SCHEMBL12874582 0.75 PLAU (0.46) PLAUDAOPOLBMEN1CYP1A2
SCHEMBL31440837 0.75 DAO (0.37) PLAUDAOALDH1A1
SCHEMBL31229804 0.75 CHRNB2 (0.31) ALDH1A1
SCHEMBL8969662 0.75 PLAU (0.41) PLAUDAOHTTALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20250100981-A1 Cis-substituted 5-(hydroxymethyl)morpholine-2-carboxamides as agonists of SSTR4 BOEHRINGER INGELHEIM INT (DE) 2025-03-27 US disclosed
WO-2025027049-A1 (2S,5R)-5-(HYDROXYMETHYL)MORPHOLINE-2-CARBOXAMIDES AS AGONISTS OF SSTR4 BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2025-02-06 WO disclosed
WO-2020061146-A1 PREPARATION OF HALOGEN ANALOGS OF PICLORAM DOW AGROSCIENCES LLC (US) 2020-03-26 WO disclosed
EP-3099672-A1 FUSED IMIDAZOLE COMPOUNDS ONO Pharmaceutical Co., Ltd. (JP) 2016-12-07 EP disclosed
WO-2015115673-A1 FUSED IMIDAZOLE COMPOUNDS ONO PHARMACEUTICAL CO., LTD. (JP) 2015-08-06 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20250100981-A1 Cis-substituted 5-(hydroxymethyl)morpholine-2-carboxamides as agonists of SSTR4 SSTR4, SSTR5, SSTR2 PLAU 2989/4885DAO 3013/4885POLB 4623/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.