SCHEMBL1698255

SCHEMBL1698255

O=C(O)c1nn(-c2cccc(C(F)(F)F)c2)c(=O)cc1O

nearest known ligand 0.68

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.68
KDM4E B2RXH2 1/20 0.68
POLB P06746 3/20 0.65
KMT2A Q03164 9/20 0.55
GAA P10253 4/20 0.53
MEN1 O00255 5/20 0.53
SMN1; SMN2 Q16637 4/20 0.53
MAPT P10636 4/20 0.53
TDP1 Q9NUW8 1/20 0.53
L3MBTL1 Q9Y468 1/20 0.53
FHIT P49789 1/20 0.51
NPSR1 Q6W5P4 1/20 0.51
CYP1A2 P05177 2/20 0.50
CYP2C9 P11712 2/20 0.50
CYP2C19 P33261 2/20 0.50
LMNA P02545 2/20 0.50
CYP3A4 P08684 1/20 0.50
HPGD P15428 1/20 0.50
ALKBH5 Q6P6C2 1/20 0.50
RAB9A P51151 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1750835 0.82 KMT2A (0.77) ALDH1A1KDM4EKMT2AGAAMEN1
SCHEMBL4483384 0.79 POLB (0.63) ALDH1A1POLBKMT2AMEN1MAPT
SCHEMBL9184563 0.79 POLB (1.00) POLBKMT2AMAPK1
SCHEMBL11519772 0.77 KMT2A (0.55) ALDH1A1POLBKMT2AGAAMEN1
SCHEMBL11274830 0.76 KMT2A (0.55) ALDH1A1POLBKMT2AGAAMEN1
SCHEMBL16569044 0.76 POLB (0.54) ALDH1A1POLBKMT2AMEN1MAPT
SCHEMBL518434 0.76 KMT2A (0.61) ALDH1A1POLBKMT2AGAAMEN1
SCHEMBL28734569 0.75 ALDH1A1 (0.74) ALDH1A1KDM4EKMT2AGAAMEN1
SCHEMBL519301 0.75 CYP1A2 (0.63) ALDH1A1POLBKMT2AGAAMEN1
SCHEMBL518604 0.74 KMT2A (0.67) ALDH1A1POLBKMT2AGAAMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011160189-A1 METHOD OF SCREENING FOR INHIBITORS OF sPLA2-IIA SCOTT KIERAN (AU) 2011-12-29 WO disclosed
WO-2011160189-A1 METHOD OF SCREENING FOR INHIBITORS OF sPLA2-IIA SCOTT KIERAN (AU) 2011-12-29 WO disclosed
EP-1091958-A1 SALTS OF PAROXETINE SMITHKLINE BEECHAM PLC (GB) 2001-04-18 EP disclosed
WO-2000001692-A1 SALTS OF PAROXETINE SMITHKLINE BEECHAM PLC (GB) 2000-01-13 WO disclosed