SCHEMBL169902

SCHEMBL169902

C=CC(=O)Nc1cn[nH]c1

nearest known ligand 0.49

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
TGM2 P21980 11/20 0.48
PIM1 P11309 1/20 0.46
PIM3 Q86V86 1/20 0.46
PIM2 Q9P1W9 1/20 0.46
F13A1 P00488 1/20 0.46
LMNA P02545 1/20 0.46
TGM1 P22735 1/20 0.46
TGM3 Q08188 1/20 0.46
KDM1A O60341 1/20 0.41
MAOA P21397 1/20 0.41
BTK Q06187 4/20 0.39
ITK Q08881 2/20 0.39
MTOR P42345 1/20 0.38
BLK P51451 1/20 0.38
BMX P51813 1/20 0.38
JAK3 P52333 1/20 0.38
MAPK7 Q13164 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2898099 0.76
SCHEMBL929848 0.76 PIM1 (0.51) PIM1PIM3PIM2LMNAKDM1A
SCHEMBL28534540 0.75 TGM2 (0.56) TGM2F13A1LMNATGM1TGM3
SCHEMBL4158764 0.75
SCHEMBL929849 0.75 PIM1 (0.50) PIM1PIM3PIM2KDM1AMAOA
Hydrochloric Acid SCHEMBL20557184 0.73 PIM1 (0.49) PIM1PIM3PIM2LMNAKDM1A
SCHEMBL17159814 0.72 PIM1 (0.69) PIM1PIM3PIM2LMNAKDM1A
SCHEMBL21585659 0.71 TGM2 (0.55) TGM2F13A1LMNATGM1TGM3
SCHEMBL439369 0.71 TGM2 (0.79) TGM2F13A1LMNATGM1TGM3
SCHEMBL16053417 0.71 TGM2 (0.64) TGM2F13A1LMNATGM1TGM3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023227125-A1 NEW FUSED-HETEROCYCLIC COMPOUND AS CDK INHIBITOR AND USE THEREOF 杭州德睿智药科技有限公司 2023-11-30 WO disclosed
EP-2424368-A1 PYRROLOTRIAZINE COMPOUNDS Locus Pharmaceuticals, Inc. (US) 2012-03-07 EP disclosed
WO-2010126960-A1 PYRROLOTRIAZINE COMPOUNDS LOCUS PHARMACEUTICALS, INC. (US) 2010-11-04 WO disclosed