SCHEMBL17004207

SCHEMBL17004207

c1cc2cc(-c3ccc(OC4C5CC6CC4CN(C6)C5)nn3)ccc2[nH]1

nearest known ligand 0.64

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CHRNA7 P36544 14/20 0.64
CHRNB2 P17787 7/20 0.55
CHRNA4 P43681 7/20 0.55
CHRNB4 P30926 6/20 0.55
CHRNA3 P32297 6/20 0.55
KCNH2 Q12809 6/20 0.46
HTR3A P46098 1/20 0.42
DYRK3 O43781 1/20 0.35
CCNT1 O60563 1/20 0.35
CDK9 P50750 1/20 0.35
CDK5 Q00535 1/20 0.35
DYRK1A Q13627 1/20 0.35
CDK5R1 Q15078 1/20 0.35
DYRK2 Q92630 1/20 0.35
DYRK1B Q9Y463 1/20 0.35
HTT P42858 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29604852 1.00 CHRNA7 (0.64) CHRNA7CHRNB2CHRNA4CHRNB4CHRNA3
SCHEMBL17004212 0.85 CHRNA7 (0.56) CHRNA7CHRNB2CHRNA4CHRNB4CHRNA3
SCHEMBL29604064 0.82 KCNH2 (0.47) CHRNA7CHRNB2CHRNA4CHRNB4CHRNA3
SCHEMBL17004276 0.82 KCNH2 (0.47) CHRNA7CHRNB2CHRNA4CHRNB4CHRNA3
SCHEMBL17004229 0.80 CHRNA7 (0.48) CHRNA7CHRNB2CHRNA4CHRNB4CHRNA3
SCHEMBL29604864 0.80 CHRNA7 (0.47) CHRNA7CHRNB2CHRNA4CHRNB4CHRNA3
SCHEMBL17004358 0.79 CHRNA7 (0.56) CHRNA7CHRNB2CHRNA4CHRNB4CHRNA3
Abt-107 SCHEMBL31393053 0.78 CHRNA7 (1.00) CHRNA7CHRNB2CHRNA4CHRNB4CHRNA3
Abt-107 SCHEMBL373047 0.78 CHRNA7 (1.00) CHRNA7CHRNB2CHRNA4CHRNB4CHRNA3
Abt-107 SCHEMBL1542259 0.78 CHRNA7 (1.00) CHRNA7CHRNB2CHRNA4CHRNB4CHRNA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2099795-B1 AZAADAMANTANE DERIVATIVES AND THEIR USES AS NICOTINIC ACETYLCHOLINE RECEPTORS LIGANDS ABBVIE BAHAMAS LTD (BS) 2015-08-19 EP disclosed