SCHEMBL17004352

SCHEMBL17004352

N#Cc1ccccc1-c1cccc2c(OCC3CCNCC3)c(-c3cccs3)c(=O)[nH]c12

nearest known ligand 0.52

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
PDE2A O00408 6/20 0.52
PIM1 P11309 2/20 0.37
PLAT P00750 3/20 0.34
HDAC3 O15379 1/20 0.34
HDAC1 Q13547 1/20 0.34
HDAC2 Q92769 1/20 0.34
KDM4E B2RXH2 2/20 0.33
CCNA2 P20248 1/20 0.32
CDK2 P24941 1/20 0.32
CCNA1 P78396 1/20 0.32
SYK P43405 2/20 0.32
KDM1A O60341 1/20 0.32
MAOB P27338 1/20 0.32
SLC6A2 P23975 2/20 0.32
SLC6A4 P31645 2/20 0.32
SLC6A3 Q01959 1/20 0.32
HTR3A P46098 1/20 0.31
KCNH2 Q12809 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17004307 0.93 PDE2A (0.55) PDE2APIM1PLATHDAC3HDAC1
SCHEMBL17004318 0.89 PDE2A (0.51) PDE2AHDAC3HDAC1HDAC2CCNA2
SCHEMBL17004349 0.86 PDE2A (0.54) PDE2APLATHDAC3HDAC1HDAC2
SCHEMBL17004334 0.85 PDE2A (0.57) PDE2AHDAC3HDAC1HDAC2CCNA2
SCHEMBL17004302 0.84 PDE2A (0.50) PDE2AHDAC3HDAC1HDAC2KDM1A
SCHEMBL935940 0.84 PDE2A (0.62) PDE2APIM1HDAC3HDAC1HDAC2
SCHEMBL17004360 0.83 PDE2A (0.55) PDE2APLATHDAC3HDAC1HDAC2
SCHEMBL17004369 0.83 PDE2A (0.51) PDE2AHDAC3HDAC1HDAC2KDM1A
SCHEMBL17004310 0.82 PDE2A (0.62) PDE2APIM1PLATHDAC3HDAC1
SCHEMBL937313 0.81 PDE2A (0.64) PDE2AHDAC3HDAC1HDAC2CCNA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2456440-B1 QUINOLINONE PDE2 INHIBITORS MERCK SHARP & DOHME (US) 2015-08-19 EP claimed