SCHEMBL17004641

SCHEMBL17004641

COc1ccc(-c2cc(-c3ccc(C4CN(C=O)CCO4)cc3)cnc2N)cn1

nearest known ligand 0.51

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 5/20 0.51
FYN P06241 9/20 0.44
MAP4K4 O95819 2/20 0.39
CHEK2 O96017 1/20 0.39
TGFBR1 P36897 4/20 0.39
ACVR1 Q04771 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16672245 0.84 CHEK2 (0.55) FYNMAP4K4CHEK2
SCHEMBL17004633 0.82 KCNH2 (0.53) KCNH2MAP4K4
SCHEMBL19086089 0.78 LRRK2 (0.60)
SCHEMBL13837101 0.77 KCNH2 (0.59) KCNH2FYNMAP4K4CHEK2TGFBR1
SCHEMBL17004628 0.73 FYN (0.73) KCNH2FYNTGFBR1ACVR1
SCHEMBL13837178 0.72 KCNH2 (0.70) KCNH2FYNMAP4K4CHEK2TGFBR1
SCHEMBL2226033 0.72 FYN (0.76) KCNH2FYNMAP4K4CHEK2TGFBR1
SCHEMBL16530537 0.72 JAK2 (0.59)
SCHEMBL12518229 0.71 KCNH2 (0.79) KCNH2FYNMAP4K4CHEK2TGFBR1
SCHEMBL19086085 0.70 LRRK2 (0.59)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2526090-B1 NEW ANTI-MALARIAL AGENTS MEDICINES FOR MALARIA VENTURE MMV (CH) 2015-08-19 EP claimed