SCHEMBL17008673

SCHEMBL17008673

C[C@@H](C#N)NC(=O)[C@@H]1CCC(F)(F)C[C@H]1c1nn(-c2ncccc2F)cc1-c1ccc(N2CCS(O)(O)CC2)cc1

nearest known ligand 0.49

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
CTSK P43235 13/20 0.49
IDH1 O75874 2/20 0.33
PRKD1 Q15139 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17008671 0.95 CTSK (0.55) CTSKIDH1PRKD1
SCHEMBL17008366 0.94 CTSK (0.49) CTSKIDH1PRKD1
SCHEMBL17008382 0.93 CTSK (0.49) CTSKIDH1PRKD1
SCHEMBL17008364 0.90 CTSK (0.44) CTSKIDH1PRKD1
SCHEMBL17008802 0.89 CTSK (0.63) CTSK
SCHEMBL17008383 0.89 CTSK (0.43) CTSKIDH1PRKD1
SCHEMBL17020305 0.89 CTSK (0.54) CTSKIDH1
SCHEMBL17008674 0.88 CTSK (0.42) CTSKPRKD1
SCHEMBL18279837 0.87 CTSK (0.48) CTSKIDH1
SCHEMBL17020277 0.87 CTSK (0.48) CTSKIDH1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3104705-A1 CATHEPSIN CYSTEINE PROTEASE INHIBITORS Merck Sharp & Dohme Corp. (US) 2016-12-21 EP claimed
WO-2015123089-A1 CATHEPSIN CYSTEINE PROTEASE INHIBITORS MERCK SHARP & DOHME CORP. (US) 2015-08-20 WO claimed