SCHEMBL17008807

SCHEMBL17008807

N#CC1(NC(=O)[C@@H]2CCCC[C@H]2c2nn(-c3ccc(C(F)(F)F)cn3)cc2-c2ccc(N3CCS(O)(O)CC3)cc2)CC1

nearest known ligand 0.67

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
CTSK P43235 18/20 0.67
CTSB P07858 4/20 0.43
CTSS P25774 4/20 0.43
KCNH2 Q12809 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17008806 0.95 CTSK (0.75) CTSKCTSBCTSSKCNH2
SCHEMBL17008755 0.91 CTSK (0.60) CTSKCTSBCTSSKCNH2
SCHEMBL17008665 0.91 CTSK (0.76) CTSKCTSBCTSSKCNH2
SCHEMBL18858010 0.90 CTSK (0.67) CTSKCTSBCTSSKCNH2
SCHEMBL17020289 0.87 CTSK (0.85) CTSKCTSBCTSSKCNH2
SCHEMBL17008248 0.87 CTSK (0.69) CTSKCTSBCTSSKCNH2
SCHEMBL17008273 0.86 CTSK (0.72) CTSKCTSBCTSSKCNH2
SCHEMBL17008291 0.86 CTSK (0.68) CTSKCTSBCTSSKCNH2
SCHEMBL18279767 0.86 CTSK (0.72) CTSKCTSBCTSSKCNH2
SCHEMBL17008648 0.86 CTSK (0.72) CTSKCTSBCTSSKCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3104705-A1 CATHEPSIN CYSTEINE PROTEASE INHIBITORS Merck Sharp & Dohme Corp. (US) 2016-12-21 EP claimed
WO-2015123089-A1 CATHEPSIN CYSTEINE PROTEASE INHIBITORS MERCK SHARP & DOHME CORP. (US) 2015-08-20 WO claimed