SCHEMBL1701050

SCHEMBL1701050

O=C(O)C(O)(O)CCCc1ccccc1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 4/20 0.53
HDAC8 Q9BY41 4/20 0.53
HDAC3 O15379 3/20 0.53
HDAC2 Q92769 3/20 0.53
HDAC6 Q9UBN7 3/20 0.53
HDAC5 Q9UQL6 3/20 0.53
HDAC4 P56524 2/20 0.53
HDAC7 Q8WUI4 2/20 0.53
HDAC10 Q969S8 2/20 0.53
HDAC11 Q96DB2 2/20 0.53
HDAC9 Q9UKV0 2/20 0.53
MAPK1 P28482 1/20 0.53
ADRA1A P35348 1/20 0.53
SLC6A3 Q01959 1/20 0.53
SMN1; SMN2 Q16637 1/20 0.53
GRM2 Q14416 2/20 0.50
GRM3 Q14832 2/20 0.50
MAPT P10636 1/20 0.50
RXFP1 Q9HBX9 1/20 0.50
NPC1 O15118 2/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8662896 0.92 MAPT (0.56) HDAC1HDAC8HDAC3HDAC2HDAC6
SCHEMBL9620413 0.92 MAPT (0.56) HDAC1HDAC8HDAC3HDAC2HDAC6
SCHEMBL8666510 0.92 MAPT (0.56) HDAC1HDAC8HDAC3HDAC2HDAC6
SCHEMBL9620303 0.92 MAPT (0.56) HDAC1HDAC8HDAC3HDAC2HDAC6
SCHEMBL9098501 0.88 SLC13A5 (0.50) HDAC1HDAC8HDAC3HDAC2HDAC6
SCHEMBL28202938 0.85 LMNA (0.51) HDAC1HDAC8HDAC3HDAC2HDAC6
SCHEMBL28351862 0.82 POLB (0.53) HDAC1HDAC8HDAC3HDAC2HDAC6
SCHEMBL27605425 0.81 CES1 (0.53) HDAC1HDAC8HDAC3HDAC2HDAC6
SCHEMBL29281939 0.79 HDAC3 (0.50) HDAC1HDAC8HDAC3HDAC2HDAC6
SCHEMBL10538923 0.79 HDAC3 (0.50) HDAC1HDAC8HDAC3HDAC2HDAC6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 12 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2694577-A1 THERMOPLASTIC MOULDING COMPOSITION MADE OF POLYARYLENE ETHERS AND POLYPHENYLENE SULPHIDE WITH IMPROVED PROCESSING STABILITY BASF SE (DE) 2014-02-12 EP disclosed
EP-2576676-A1 REINFORCED THERMOPLASTIC MOLDING COMPOUNDS BASED ON POLYARYLENE ETHERS BASF SE (DE) 2013-04-10 EP disclosed
EP-2550335-A1 IMPROVED BLENDS OF POLYARYLENE ETHERS AND POLYARYLENE SULFIDES BASF SE (DE) 2013-01-30 EP disclosed
EP-2542623-A1 IMPROVED BLENDS OF POLYARYLENE ETHERS AND POLYARYLENE SULFIDES BASF SE (DE) 2013-01-09 EP disclosed
WO-2012156327-A1 THERMOPLASTIC MOULDING COMPOSITION MADE OF POLYARYLENE ETHERS AND POLYPHENYLENE SULPHIDE WITH IMPROVED PROCESSING STABILITY BASF SE (DE) 2012-11-22 WO disclosed
EP-2513193-A1 IMPROVED BLENDS OF POLYARYLENE ETHERS AND POLYARYLENE SULFIDES BASF SE (DE) 2012-10-24 EP disclosed
EP-2513191-A1 IMPROVED BLENDS OF POLYARYLENE ETHERS AND POLYARYLENE SULFIDES BASF SE (DE) 2012-10-24 EP disclosed
WO-2011147758-A1 REINFORCED THERMOPLASTIC MOLDING COMPOUNDS BASED ON POLYARYLENE ETHERS BASF SE (DE) 2011-12-01 WO disclosed
WO-2011117153-A1 IMPROVED BLENDS OF POLYARYLENE ETHERS AND POLYARYLENE SULFIDES BASF SE (DE) 2011-09-29 WO disclosed
WO-2011107389-A1 IMPROVED BLENDS OF POLYARYLENE ETHERS AND POLYARYLENE SULFIDES BASF SE (DE) 2011-09-09 WO disclosed
WO-2011073197-A1 IMPROVED BLENDS OF POLYARYLENE ETHERS AND POLYARYLENE SULFIDES BASF SE (DE) 2011-06-23 WO disclosed
WO-2011073196-A1 IMPROVED BLENDS OF POLYARYLENE ETHERS AND POLYARYLENE SULFIDES BASF SE (DE) 2011-06-23 WO disclosed