SCHEMBL17011909

SCHEMBL17011909

NC(=O)c1ccc(-c2cc(-c3ccc([SH](=O)=O)cc3)cnc2N)cc1

nearest known ligand 0.73

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
CHEK2 O96017 14/20 0.73
FYN P06241 3/20 0.73
MKNK1 Q9BUB5 1/20 0.73
MAP4K4 O95819 3/20 0.71
CHEK1 O14757 4/20 0.63

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12516852 0.90 CHEK2 (0.88) CHEK2FYNMKNK1MAP4K4CHEK1
SCHEMBL4620246 0.85 CHEK2 (1.00) CHEK2FYNMKNK1MAP4K4CHEK1
SCHEMBL18613241 0.85 FYN (1.00) CHEK2FYNMKNK1MAP4K4CHEK1
SCHEMBL13977050 0.83 CHEK2 (0.77) CHEK2FYNMKNK1MAP4K4CHEK1
SCHEMBL28051402 0.83 CHEK2 (0.68) CHEK2FYNMKNK1MAP4K4CHEK1
SCHEMBL2228006 0.82 CHEK2 (0.75) CHEK2FYNMKNK1MAP4K4CHEK1
SCHEMBL12077792 0.81 CHEK2 (0.87) CHEK2FYNMKNK1MAP4K4CHEK1
SCHEMBL2224862 0.81 CHEK2 (0.72) CHEK2FYNMKNK1MAP4K4CHEK1
SCHEMBL12078010 0.80 MAP4K4 (0.79) CHEK2FYNMKNK1MAP4K4CHEK1
SCHEMBL12078349 0.80 CHEK2 (0.72) CHEK2FYNMKNK1MAP4K4CHEK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2526090-B1 NEW ANTI-MALARIAL AGENTS MEDICINES FOR MALARIA VENTURE MMV (CH) 2015-08-19 EP disclosed