SCHEMBL17011995

SCHEMBL17011995

CC(C)NC(=O)c1cccc(C(=O)NCc2cnn(-c3cccc(C(F)F)c3)c2)n1

nearest known ligand 0.46

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ADRB2 P07550 1/20 0.46
ELANE P08246 2/20 0.43
ALDH1A1 P00352 2/20 0.40
KDM4E B2RXH2 1/20 0.40
POLB P06746 2/20 0.39
RAB9A P51151 1/20 0.39
GRIN1 Q05586 9/20 0.39
GRIN2B Q13224 9/20 0.39
RXRA P19793 8/20 0.39
NPSR1 Q6W5P4 1/20 0.38
DDT P30046 1/20 0.38
KLKB1 P03952 1/20 0.38
KLK1 P06870 1/20 0.38
MAPK1 P28482 1/20 0.37
USP2 O75604 1/20 0.37
TSHR P16473 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8211521 0.89 ADRB2 (0.57) ADRB2ALDH1A1KDM4EPOLBRAB9A
SCHEMBL8209034 0.88 ADRB2 (0.47) ADRB2ALDH1A1KDM4EPOLBNPSR1
SCHEMBL8210993 0.88 ADRB2 (0.46) ADRB2ALDH1A1KDM4EPOLBKLKB1
SCHEMBL12853254 0.88 HPGD (0.44) ADRB2ALDH1A1KDM4EPOLBRAB9A
SCHEMBL8206269 0.87 ADRB2 (0.45) ADRB2ALDH1A1KDM4EPOLBRAB9A
SCHEMBL12853297 0.87 DDT (0.53) ADRB2ELANERAB9ANPSR1DDT
SCHEMBL12853294 0.85 KDM4E (0.44) ADRB2ALDH1A1KDM4EPOLBNPSR1
SCHEMBL12853289 0.85 KCNJ1 (0.46) ADRB2ELANEALDH1A1KDM4EPOLB
SCHEMBL8205788 0.85 ADRB2 (0.43) ADRB2ALDH1A1KDM4EPOLBKLKB1
SCHEMBL12853298 0.84 ADRB2 (0.44) ADRB2ALDH1A1POLBNPSR1KLKB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2132178-B1 JNK INHIBITORS MERCK SHARP & DOHME (US) 2015-08-19 EP disclosed
US-8975389-B2 Nucleic acid chemical modifications ALNYLAM PHARMACEUTICALS, INC. (US) 2015-03-10 US disclosed