SCHEMBL170246

SCHEMBL170246

CC(CCN)=C(C(=O)O)C(C)C

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GABRR1 P24046 4/20 0.37
GABRP O00591 3/20 0.32
GABRD O14764 3/20 0.32
GABRA1 P14867 3/20 0.32
GABRB1 P18505 3/20 0.32
GABRG2 P18507 3/20 0.32
GABRB3 P28472 3/20 0.32
GABRA5 P31644 3/20 0.32
GABRA3 P34903 3/20 0.32
GABRA2 P47869 3/20 0.32
GABRB2 P47870 3/20 0.32
GABRA4 P48169 3/20 0.32
GABRE P78334 3/20 0.32
GABRA6 Q16445 3/20 0.32
GABRG1 Q8N1C3 3/20 0.32
GABRG3 Q99928 3/20 0.32
GABRQ Q9UN88 3/20 0.32
PAOX Q6QHF9 1/20 0.32
GABRR3 A8MPY1 1/20 0.31
HDAC3 O15379 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL27893185 0.98 GABRR1 (0.35) GABRR1GABRPGABRDGABRA1GABRB1
Methacrylic Acid SCHEMBL6561456 0.91 GABRR1 (0.31) GABRR1
SCHEMBL11112222 0.88 GABRR1 (0.43) GABRR1GABRPGABRDGABRA1GABRB1
SCHEMBL11767532 0.86
SCHEMBL18986068 0.80 HDAC1 (0.40) HDAC3THRBTSHRHDAC1HDAC2
SCHEMBL27838004 0.78
SCHEMBL6668764 0.77 CAMK2A (0.41)
SCHEMBL9322240 0.75 ALDH1A1 (0.36)
SCHEMBL7857868 0.72 PAOX (0.37) GABRR1GABRPGABRDGABRA1GABRB1
Hydrochloric Acid SCHEMBL7120514 0.71 ALDH1A1 (0.33)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 71 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0900563-B1 Production of pharmaceutical formulations containing aescin for treatment of edema and venous disorders KLINGE CO CHEM PHARM FAB (DE) 2004-02-11 EP claimed
WO-1999030685-A1 POLYMERIC MICROPOROUS FILM COATED SUBCUTANEOUS IMPLANTS AMERICAN HOME PRODUCTS CORPORATION (US) 1999-06-24 WO claimed
EP-3487916-B1 FUNCTIONALIZED PARTICULATE BICARBONATE AS BLOWING AGENT, FOAMABLE POLYMER COMPOSITION CONTAINING IT, AND ITS USE IN MANUFACTURING A THERMOPLASTIC FOAMED POLYMER SOLVAY (BE) 2025-09-03 EP disclosed
US-12116467-B2 Foamable crosslinkable polymer composition containing a functionalized particulate bicarbonate as blowing agent and method for manufacturing a crosslinked foamed polymer therefrom SOLVAY SA (BE) 2024-10-15 US disclosed
EP-3655469-B1 FUNCTIONALIZED PARTICULATE BICARBONATE AS BLOWING AGENT, FOAMABLE POLYMER COMPOSITION CONTAINING IT, AND ITS USE IN MANUFACTURING A THERMOPLASTIC FOAMED POLYMER SOLVAY (BE) 2024-09-25 EP disclosed
US-20240239980-A1 FUNCTIONALIZED PARTICULATE BICARBONATE AS BLOWING AGENT, FOAMABLE POLYMER COMPOSITION CONTAINING IT, AND ITS USE IN MANUFACTURING A THERMOPLASTIC FOAMED POLYMER SOLVAY SA (BE) 2024-07-18 US disclosed
US-11926722-B2 Functionalized particulate bicarbonate as blowing agent, foamable polymer composition containing it, and its use in manufacturing a thermoplastic foamed polymer SOLVAY SA (BE) 2024-03-12 US disclosed
EP-3655470-B1 FUNCTIONALIZED PARTICULATE BICARBONATE AS BLOWING AGENT, FOAMABLE POLYMER COMPOSITION CONTAINING IT, AND ITS USE IN MANUFACTURING A THERMOPLASTIC FOAMED POLYMER SOLVAY (BE) 2023-09-20 EP disclosed
US-11421094-B2 Functionalized particulate bicarbonate as blowing agent, foamable polymer composition containing it, and its use in manufacturing a thermoplastic foamed polymer SOLVAY SA (BE) 2022-08-23 US disclosed
US-20220259396-A1 FUNCTIONALIZED PARTICULATE BICARBONATE AS BLOWING AGENT, FOAMABLE POLYMER COMPOSITON CONTAINING IT, AND ITS USE IN MANUFACTURING A THERMOPLASTIC FOAMED POLYMER SOLVAY SA (BE) 2022-08-18 US disclosed
US-20220175351-A1 Devices and Methods for Collecting Gastrointestinal Samples ENVIVO BIO INC. (US) 2022-06-09 US disclosed
US-20110002906-A1 Purification and Isolation of Recombinant Oxalate Degrading Enzymes and Spray-Dried Particles Containing Oxalate Degrading Enzymes OXTHERA INTELLECTUAL PROPERTY AB (SE) 2011-01-06 US disclosed
WO-2011000523-A1 PURIFICATION AND ISOLATION OF RECOMBINANT OXALATE DEGRADING ENZYMES AND SPRAY-DRIED PARTICLES CONTAINING OXALATE DEGRADING ENZYMES OXTHERA INTELLECTUAL PROPERTY AB (SE) 2011-01-06 WO disclosed
WO-2010102218-A1 COMPOUNDS AND COMPOSITIONS FOR COGNITION-ENHANCEMENT, METHODS OF MAKING, AND METHODS OF TREATING MITHRIDION, INC. (US) 2010-09-10 WO disclosed
EP-2153834-A2 Extended release pharmaceutical compositions comprising quetiapine salts Farmaprojects, S.A. (ES) 2010-02-17 EP disclosed
US-20090324716-A1 Coated Particles Containing Pharmaceutically Active Agents JOHNSON & JOHNSON CONSUMER INC. 2009-12-31 US disclosed
WO-2009158368-A1 COATED PARTICLES CONTAINING PHARMACEUTICALLY ACTIVE AGENTS MCNEIL-PPC, INC. (US) 2009-12-30 WO disclosed
EP-1838291-A4 PHARMACEUTICAL FORMULATIONS AND METHODS OF USE PHARMANOVA INC (US) 2008-12-03 EP disclosed
EP-1838291-A2 PHARMACEUTICAL FORMULATIONS AND METHODS OF USE Pharmanova Inc. (US) 2007-10-03 EP disclosed
WO-2006078811-A2 PHARMACEUTICAL FORMULATIONS AND METHODS OF USE PHARMANOVA INC. (US) 2006-07-27 WO disclosed