SCHEMBL1703240

SCHEMBL1703240

N#Cc1c(Cl)ccnc1-c1ccc(NC(=O)Nc2cc(F)cc(F)c2)cc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDR P35968 10/20 0.45
LMNA P02545 2/20 0.41
MAPT P10636 2/20 0.41
MEN1 O00255 1/20 0.41
KMT2A Q03164 1/20 0.41
RIPK1 Q13546 1/20 0.40
PPARG P37231 1/20 0.40
PDGFRA P16234 1/20 0.40
MET P08581 2/20 0.39
RAB9A P51151 3/20 0.39
NPC1 O15118 2/20 0.39
SMN1; SMN2 Q16637 2/20 0.39
TP53 P04637 1/20 0.39
TSHR P16473 1/20 0.39
HTT P42858 1/20 0.39
NLRP3 Q96P20 1/20 0.39
KIT P10721 1/20 0.39
AURKA O14965 1/20 0.39
ROCK2 O75116 1/20 0.39
RPS6KA5 O75582 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3443775 0.90 KDR (0.50) KDRLMNAMAPTMEN1KMT2A
SCHEMBL3442309 0.88 MEN1 (0.57) KDRLMNAMAPTMEN1KMT2A
SCHEMBL1704022 0.86 KDR (0.53) KDRMEN1KMT2AMETKIT
SCHEMBL3442391 0.85 KDR (0.56) KDRLMNAMAPTMEN1KMT2A
SCHEMBL12346315 0.83 ALDH1A1 (0.47) KDRLMNAMAPTMETTSHR
SCHEMBL3442732 0.83 KDR (0.57) KDRLMNAMAPTMEN1KMT2A
SCHEMBL3443115 0.83 KDR (0.53) KDRRIPK1KITLCKLYN
SCHEMBL1702775 0.82 KDR (0.58) KDRMAPTPDGFRARAB9ANPC1
SCHEMBL1703220 0.82 KDR (0.53) KDRRIPK1PDGFRAMETRAB9A
SCHEMBL3443455 0.81 CNR1 (0.52) KDRKMT2APDGFRAMETSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1807424-B1 NOVEL KINASE INHIBITORS ABBOTT LAB (US) 2012-04-18 EP disclosed
US-7812166-B2 Kinase inhibitors ABBOTT LABORATORIES (US) 2010-10-12 US disclosed
US-20060178378-A1 Novel kinase inhibitors ABBVIE INC. 2006-08-10 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20060178378-A1 Novel kinase inhibitors ABL1, MAP3K19, MAP3K20 KDR 434/4885LMNA 4320/4885MAPT 2564/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.