SCHEMBL1704154

SCHEMBL1704154

C[C@H]1CN(Cc2ccc(CC(=O)N3CCC(Nc4cccc(F)c4)CC3)cc2)CCN1C(=O)OCc1ccccc1

nearest known ligand 0.65

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
MLNR O43193 19/20 0.65
CYP3A4 P08684 6/20 0.65
CYP2D6 P10635 1/20 0.65
KCNH2 Q12809 1/20 0.65

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1704527 1.00 MLNR (0.65) MLNRCYP3A4CYP2D6KCNH2
SCHEMBL4175748 0.89 MLNR (0.73) MLNRCYP3A4CYP2D6KCNH2
SCHEMBL4187464 0.89 MLNR (0.73) MLNRCYP3A4CYP2D6KCNH2
SCHEMBL1704165 0.88 MLNR (0.67) MLNRCYP3A4CYP2D6KCNH2
SCHEMBL1703977 0.85 MLNR (0.64) MLNRCYP3A4CYP2D6KCNH2
SCHEMBL1704593 0.84 MLNR (0.46) MLNRCYP3A4CYP2D6KCNH2
SCHEMBL4188248 0.81 MLNR (0.75) MLNRCYP3A4CYP2D6KCNH2
SCHEMBL1705080 0.80 MLNR (0.70) MLNRCYP3A4CYP2D6KCNH2
SCHEMBL4185723 0.80 MLNR (0.76) MLNRCYP3A4CYP2D6KCNH2
Camicinal SCHEMBL1703910 0.79 MLNR (1.00) MLNRCYP3A4CYP2D6KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2441763-A1 Benzylpiperazine derivatives useful for the treatment of gastrointestinal disorders Glaxo Group Limited (GB) 2012-04-18 EP disclosed