SCHEMBL1703977

SCHEMBL1703977

C[C@H]1CN(Cc2ccc(CCC(=O)N3CCC(Nc4ccc(F)cc4)CC3)cc2)CCN1C(=O)OCc1ccccc1

nearest known ligand 0.64

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
MLNR O43193 15/20 0.64
CYP3A4 P08684 7/20 0.54
PDK1 Q15118 1/20 0.46
PDK2 Q15119 1/20 0.46
PDK3 Q15120 1/20 0.46
PDK4 Q16654 1/20 0.46
CCR1 P32246 2/20 0.45
CYP2D6 P10635 1/20 0.45
KCNH2 Q12809 1/20 0.45
YAP1 P46937 1/20 0.44
MEN1 O00255 1/20 0.44
KMT2A Q03164 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4185674 0.88 MLNR (0.73) MLNRCYP3A4CCR1CYP2D6KCNH2
SCHEMBL1704527 0.85 MLNR (0.65) MLNRCYP3A4CYP2D6KCNH2
SCHEMBL1704154 0.85 MLNR (0.65) MLNRCYP3A4CYP2D6KCNH2
SCHEMBL4183557 0.82 MLNR (0.77) MLNRCYP3A4CYP2D6KCNH2
SCHEMBL4597349 0.79 MLNR (0.70) MLNRCYP3A4CYP2D6KCNH2
SCHEMBL1703823 0.79 MLNR (0.70) MLNRCYP3A4CYP2D6KCNH2
SCHEMBL1704131 0.78 MLNR (1.00) MLNRCYP3A4CYP2D6KCNH2
SCHEMBL14646619 0.78 PDK1 (0.59) PDK1PDK2PDK3PDK4CCR1
SCHEMBL1704619 0.78 MLNR (1.00) MLNRCYP3A4CYP2D6KCNH2
SCHEMBL2010214 0.77 MLNR (0.46) MLNRCYP3A4PDK1PDK2PDK3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2441763-A1 Benzylpiperazine derivatives useful for the treatment of gastrointestinal disorders Glaxo Group Limited (GB) 2012-04-18 EP disclosed