SCHEMBL1705330

SCHEMBL1705330

CC(C)c1nccc2cc(O[C@H]3CC[C@@H](N)CC3)ccc12

nearest known ligand 0.51

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ROCK1 Q13464 13/20 0.51
ROCK2 O75116 3/20 0.45
KCNH2 Q12809 2/20 0.45
IKBKB O14920 1/20 0.40
PRKACA P17612 1/20 0.36
PRKCD Q05655 1/20 0.36
PRKG1 Q13976 1/20 0.36
PKN1 Q16512 1/20 0.36
PKN2 Q16513 1/20 0.36
AAK1 Q2M2I8 1/20 0.36
CDC42BPA Q5VT25 1/20 0.36
Q6ZSR9 Q6ZSR9 1/20 0.36
BMP2K Q9NSY1 1/20 0.36
CDC42BPB Q9Y5S2 1/20 0.36
PRKCZ Q05513 1/20 0.34
LNPEP Q9UIQ6 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1706232 0.82 ROCK1 (0.48) ROCK1ROCK2KCNH2IKBKBLNPEP
SCHEMBL1204558 0.82 ROCK1 (0.74) ROCK1ROCK2KCNH2IKBKBPRKACA
SCHEMBL1204561 0.82 ROCK1 (0.74) ROCK1ROCK2KCNH2IKBKBPRKACA
SCHEMBL3113476 0.82 ROCK1 (0.74) ROCK1ROCK2KCNH2IKBKBPRKACA
SCHEMBL2337348 0.81 ROCK1 (0.54) ROCK1ROCK2KCNH2IKBKBPRKACA
SCHEMBL2337345 0.81 ROCK1 (0.54) ROCK1ROCK2KCNH2IKBKBPRKACA
SCHEMBL12211290 0.81 ROCK1 (0.54) ROCK1ROCK2KCNH2IKBKBPRKACA
SCHEMBL13757491 0.75 ROCK1 (0.51) ROCK1ROCK2KCNH2IKBKB
SCHEMBL25873194 0.75 DYRK1A (0.48) ROCK1
SCHEMBL13763597 0.73 ROCK1 (0.54) ROCK1ROCK2KCNH2IKBKBPRKACA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2125746-B1 CYCLOALKYLAMINE SUBSTITUTED ISOQUINOLINE DERIVATIVES SANOFI SA (FR) 2012-04-18 EP claimed