SCHEMBL17057151

SCHEMBL17057151

CCC(=O)c1c(Cl)cc(O)cc1Cl

nearest known ligand 0.63

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 6/20 0.63
MEN1 O00255 3/20 0.63
KMT2A Q03164 3/20 0.63
PTGS1 P23219 1/20 0.63
DRD3 P35462 1/20 0.63
HSP90AB1 P08238 1/20 0.42
HPGD P15428 3/20 0.42
CRHBP P24387 1/20 0.42
CRHR2 Q13324 1/20 0.42
HSD17B10 Q99714 1/20 0.42
MAPT P10636 1/20 0.42
MAPK1 P28482 1/20 0.42
PIK3CA P42336 1/20 0.42
NR1H2 P55055 1/20 0.38
NR1H3 Q13133 1/20 0.38
TSHR P16473 2/20 0.37
HMGCR P04035 1/20 0.36
THRB P10828 1/20 0.36
CA9 Q16790 2/20 0.35
CA12 O43570 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11217214 0.84 KMT2A (0.48) CYP3A4MEN1KMT2APTGS1DRD3
SCHEMBL23979141 0.83 CYP3A4 (0.47) CYP3A4MEN1KMT2APTGS1DRD3
SCHEMBL17056905 0.83 TSHR (0.53) CYP3A4MEN1KMT2APTGS1DRD3
SCHEMBL28154597 0.78 KMT2A (0.49) CYP3A4MEN1KMT2APTGS1DRD3
SCHEMBL27712795 0.78 HSP90AB1 (0.47) CYP3A4MEN1KMT2APTGS1DRD3
Flopropione SCHEMBL26316 0.77 CYP3A4 (1.00) CYP3A4MEN1KMT2APTGS1DRD3
SCHEMBL8239577 0.76 FEN1 (0.57) CYP3A4MEN1KMT2APTGS1DRD3
SCHEMBL7300081 0.76 MEN1 (0.65) CYP3A4MEN1KMT2APTGS1DRD3
SCHEMBL28155500 0.76 CYP3A4 (0.65) CYP3A4MEN1KMT2APTGS1DRD3
SCHEMBL16284311 0.74 CYP3A4 (0.63) CYP3A4MEN1KMT2APTGS1DRD3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015129926-A1 PYRAZOLE AMIDE DERIVATIVE TEIJIN PHARMA LIMITED (JP) 2015-09-03 WO disclosed