SCHEMBL17059593

SCHEMBL17059593

COc1cc(NCCN(C)C)ccc1[N+](=O)[O-]

nearest known ligand 0.50

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 8/20 0.50
GAA P10253 3/20 0.50
MAPT P10636 3/20 0.50
MAPK1 P28482 2/20 0.50
KDM4E B2RXH2 1/20 0.50
L3MBTL1 Q9Y468 1/20 0.50
NPSR1 Q6W5P4 1/20 0.50
PKM P14618 1/20 0.44
TMEM97 Q5BJF2 4/20 0.43
LMNA P02545 2/20 0.43
TDP1 Q9NUW8 1/20 0.43
MEN1 O00255 1/20 0.42
KMT2A Q03164 1/20 0.42
RAD52 P43351 1/20 0.42
POLB P06746 2/20 0.42
HTT P42858 2/20 0.41
SIRT6 Q8N6T7 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4535542 0.83 ALDH1A1 (0.52) ALDH1A1GAAMAPTMAPK1KDM4E
SCHEMBL10654179 0.83 MAPT (0.55) ALDH1A1GAAMAPTMAPK1KDM4E
SCHEMBL29588009 0.83 ALDH1A1 (0.52) ALDH1A1GAAMAPTMAPK1KDM4E
SCHEMBL29588016 0.83 ALDH1A1 (0.52) ALDH1A1GAAMAPTMAPK1KDM4E
SCHEMBL13393628 0.82 MAPT (0.44) ALDH1A1GAAMAPTMAPK1KDM4E
SCHEMBL13832433 0.82 ALDH1A1 (0.51) ALDH1A1GAAMAPTMAPK1KDM4E
SCHEMBL20718866 0.81 ALDH1A1 (0.56) ALDH1A1GAAMAPTMAPK1KDM4E
SCHEMBL14243000 0.81 NPC1 (0.52) ALDH1A1GAAMAPTMAPK1KDM4E
SCHEMBL14906663 0.81 ALDH1A1 (0.52) ALDH1A1GAAMAPTMAPK1L3MBTL1
SCHEMBL14243555 0.80 ALDH1A1 (0.49) ALDH1A1GAAMAPTMAPK1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015127873-A1 ARYLAMINO PYRAMIDINE COMPOUND AND APPLICATION THEREOF, AND PHARMACEUTICAL COMPOSITIONS AND PHARMACEUTICALLY ACCEPTABLE COMPOSITIONS PREPARED THEREFROM 上海海雁医药科技有限公司 2015-09-03 WO disclosed