SCHEMBL17059604

SCHEMBL17059604

C=CC(=O)Nc1cccc(NC(=O)Nc2ccnc(Nc3ccc(N4CCCCC4)cc3)n2)c1

nearest known ligand 0.85

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
EGFR P00533 18/20 0.85
JAK2 O60674 1/20 0.62
JAK1 P23458 1/20 0.62
TYK2 P29597 1/20 0.62
JAK3 P52333 1/20 0.62
BLK P51451 3/20 0.59
FLT3 P36888 2/20 0.59
ITK Q08881 2/20 0.57
SRC P12931 1/20 0.57
BTK Q06187 1/20 0.57

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17059694 0.92 EGFR (1.00) EGFRJAK2JAK1TYK2JAK3
SCHEMBL17059685 0.91 EGFR (1.00) EGFRJAK2JAK1TYK2JAK3
SCHEMBL17059610 0.86 EGFR (0.64) EGFRJAK2JAK1TYK2JAK3
SCHEMBL17059659 0.86 EGFR (0.87) EGFRJAK3
SCHEMBL17059692 0.84 EGFR (0.77) EGFRITKBTK
SCHEMBL17059708 0.84 EGFR (0.77) EGFRBLKFLT3ITK
SCHEMBL17059589 0.84 EGFR (0.80) EGFRITKBTK
SCHEMBL10127802 0.84 EGFR (0.87) EGFRJAK2JAK1TYK2JAK3
SCHEMBL17059592 0.84 EGFR (0.84) EGFRJAK2JAK1TYK2JAK3
SCHEMBL17059603 0.83 EGFR (0.60) EGFRJAK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015127873-A1 ARYLAMINO PYRAMIDINE COMPOUND AND APPLICATION THEREOF, AND PHARMACEUTICAL COMPOSITIONS AND PHARMACEUTICALLY ACCEPTABLE COMPOSITIONS PREPARED THEREFROM 上海海雁医药科技有限公司 2015-09-03 WO disclosed