SCHEMBL17059708

SCHEMBL17059708

C=CC(=O)Nc1cccc(NC(=O)Nc2ccnc(Nc3ccc(Cl)cc3)n2)c1

nearest known ligand 0.77

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
EGFR P00533 18/20 0.77
ITK Q08881 1/20 0.63
FLT3 P36888 1/20 0.53
BLK P51451 1/20 0.53
KDR P35968 1/20 0.53
TEK Q02763 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17059589 0.90 EGFR (0.80) EGFRITK
SCHEMBL17059692 0.90 EGFR (0.77) EGFRITK
SCHEMBL17059660 0.89 EGFR (0.68) EGFRITK
SCHEMBL17059596 0.87 EGFR (1.00) EGFRITK
SCHEMBL17059638 0.85 EGFR (0.82) EGFRITK
SCHEMBL17059604 0.84 EGFR (0.85) EGFRITKFLT3BLK
SCHEMBL17059588 0.83 EGFR (0.61) EGFRITKKDRTEK
SCHEMBL17059694 0.83 EGFR (1.00) EGFRFLT3BLK
SCHEMBL17059677 0.83 EGFR (1.00) EGFRITK
SCHEMBL14791186 0.82 ITK (0.81) EGFRITKBLK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015127873-A1 ARYLAMINO PYRAMIDINE COMPOUND AND APPLICATION THEREOF, AND PHARMACEUTICAL COMPOSITIONS AND PHARMACEUTICALLY ACCEPTABLE COMPOSITIONS PREPARED THEREFROM 上海海雁医药科技有限公司 2015-09-03 WO disclosed