SCHEMBL17059641

SCHEMBL17059641

Nc1cccc(NC(=O)Nc2ccnc(Nc3ccc(OCc4cccc(F)c4)c(Cl)c3)n2)c1

nearest known ligand 0.55

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
EGFR P00533 18/20 0.55
ERBB2 P04626 16/20 0.55
ERBB4 Q15303 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17059626 0.88 EGFR (0.62) EGFRERBB2ERBB4
SCHEMBL17059649 0.88 EGFR (0.57) EGFRERBB2ERBB4
SCHEMBL17059658 0.83 CSNK1A1 (0.58) EGFR
SCHEMBL691455 0.78 EGFR (0.78) EGFRERBB2ERBB4
SCHEMBL28771965 0.74 EGFR (0.82) EGFRERBB2ERBB4
SCHEMBL18788863 0.73 EGFR (0.61) EGFRERBB2ERBB4
SCHEMBL3505411 0.72 EGFR (0.62) EGFRERBB2ERBB4
SCHEMBL17059600 0.71 EGFR (0.74) EGFR
SCHEMBL1094554 0.71 EGFR (0.81) EGFRERBB2ERBB4
SCHEMBL691623 0.71 EGFR (0.82) EGFRERBB2ERBB4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015127873-A1 ARYLAMINO PYRAMIDINE COMPOUND AND APPLICATION THEREOF, AND PHARMACEUTICAL COMPOSITIONS AND PHARMACEUTICALLY ACCEPTABLE COMPOSITIONS PREPARED THEREFROM 上海海雁医药科技有限公司 2015-09-03 WO disclosed