SCHEMBL1706416

SCHEMBL1706416

CCCC(Cl)(Cl)CC(=O)O

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HMGCR P04035 1/20 0.40
CHRM1 P11229 1/20 0.40
TBXA2R P21731 1/20 0.40
ADRA1A P35348 1/20 0.40
TDP1 Q9NUW8 3/20 0.39
FFAR1 O14842 2/20 0.39
CPT2 P23786 1/20 0.39
TSHR P16473 4/20 0.39
CYP2D6 P10635 1/20 0.39
CYP2C19 P33261 1/20 0.39
HIF1A Q16665 1/20 0.39
FFAR3 O14843 2/20 0.38
HDAC3 O15379 1/20 0.38
HDAC1 Q13547 1/20 0.38
HDAC2 Q92769 1/20 0.38
HDAC8 Q9BY41 1/20 0.38
ALDH1A1 P00352 3/20 0.35
KDM4E B2RXH2 1/20 0.34
FDPS P14324 1/20 0.34
AKR1B1 P15121 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8789070 0.82 TDP1 (0.48) TDP1FFAR1CPT2TSHRALDH1A1
SCHEMBL8085003 0.82 TDP1 (0.48) TDP1FFAR1CPT2TSHRALDH1A1
SCHEMBL1078361 0.80 ALDH1A1 (0.36) TDP1TSHRALDH1A1FDPSHSD17B10
SCHEMBL1454489 0.79
SCHEMBL1132535 0.78 HMGCR (0.44) HMGCRCHRM1TBXA2RADRA1ATDP1
SCHEMBL2706813 0.78 ALDH1A1 (0.45) HMGCRCHRM1TBXA2RADRA1ATDP1
SCHEMBL2652438 0.77 ALDH1A1 (0.36) HMGCRCHRM1TBXA2RADRA1ATDP1
SCHEMBL9620491 0.77 FFAR1 (0.52) HMGCRCHRM1TBXA2RADRA1ATDP1
Methyl Alcohol SCHEMBL3697711 0.77 HMGCR (0.42) HMGCRCHRM1TBXA2RADRA1ATDP1
SCHEMBL10940999 0.77 HMGCR (0.48) HMGCRCHRM1TBXA2RADRA1ATDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-107898775-A IBC2 compounds are preparing the application in preventing and treating bladder cancer drug 李翀 2018-04-13 CN claimed
CN-107898775-A IBC2 compounds are preparing the application in preventing and treating bladder cancer drug 李翀 2018-04-13 CN disclosed
US-9283199-B2 Halogenated aliphatic carboxylic acids, oligomers and/or polymers thereof and their use in devitalizing external and internal neoplasms CIMAS LIMITED (CY) 2016-03-15 US disclosed
US-20160067198-A1 HALOGENATED ALIPHATIC CARBOXYLIC ACIDS, OLIGOMERS AND/OR POLYMERS THEREOF AND THEIR USE IN DEVITALIZING EXTERNAL AND INTERNAL NEOPLASMS CIMAS LIMITED (CY) 2016-03-10 US disclosed
CN-102695503-A Halogenated aliphatic carboxylic acids, oligomers and/or polymers thereof and their use for inactivating external and internal neoplasias MARDI MEDICINES LTD 2012-09-26 CN disclosed
EP-2440198-A2 HALOGENATED ALIPHATIC CARBOXYLIC ACIDS, OLIGOMERS AND/OR POLYMERS THEREOF AND THEIR USE IN DEVITALIZING EXTERNAL AND INTERNAL NEOPLASMS Mardi Medicines Ltd. (IL) 2012-04-18 EP disclosed
US-20110052641-A1 HALOGENATED ALIPHATIC CARBOXYLIC ACIDS, OLIGOMERS AND/OR POLYMERS THEREOF AND THEIR USE IN DEVITALIZING EXTERNAL AND INTERNAL NEOPLASMS MARDI MEDICINES LTD. (IL) 2011-03-03 US disclosed
WO-2010143188-A2 HALOGENATED ALIPHATIC CARBOXYLIC ACIDS, OLIGOMERS AND/OR POLYMERS THEREOF AND THEIR USE IN DEVITALIZING EXTERNAL AND INTERNAL NEOPLASMS MARDI MEDICINES LTD. (IL) 2010-12-16 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20160067198-A1 HALOGENATED ALIPHATIC CARBOXYLIC ACIDS, OLIGOMERS AND/OR POLYMERS THEREOF AND THEIR USE IN DEVITALIZING EXTERNAL AND INTERNAL NEOPLASMS CCR10, PBK, CCR3 HMGCR 3373/4885CHRM1 2072/4885TBXA2R 2987/4885
US-20110052641-A1 HALOGENATED ALIPHATIC CARBOXYLIC ACIDS, OLIGOMERS AND/OR POLYMERS THEREOF AND THEIR USE IN DEVITALIZING EXTERNAL AND INTERNAL NEOPLASMS CCR10, PBK, CCR3 HMGCR 3373/4885CHRM1 2072/4885TBXA2R 2987/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.