SCHEMBL17065975

SCHEMBL17065975

COCCC(=O)Nc1cn2cc(Br)ccc2n1

nearest known ligand 0.57

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
MAP3K5 Q99683 7/20 0.57
ROCK2 O75116 1/20 0.45
PIK3CA P42336 4/20 0.44
KDM4E B2RXH2 1/20 0.39
NPC1 O15118 1/20 0.39
ALDH1A1 P00352 1/20 0.39
POLB P06746 1/20 0.39
GAA P10253 1/20 0.39
RAB9A P51151 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
PIK3CG P48736 1/20 0.39
MAPK8 P45983 1/20 0.39
MAPK10 P53779 1/20 0.39
ABL1 P00519 1/20 0.38
LRRK2 Q5S007 1/20 0.38
HPGD P15428 1/20 0.38
TSHR P16473 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17065980 0.87 MAP3K5 (0.56) MAP3K5ROCK2PIK3CAKDM4ENPC1
SCHEMBL17065991 0.80 MAP3K5 (0.56) MAP3K5ROCK2PIK3CAKDM4ENPC1
SCHEMBL31286840 0.80 MAP3K5 (0.56) MAP3K5ROCK2KDM4ENPC1ALDH1A1
SCHEMBL2947671 0.78 MAP3K5 (0.64) MAP3K5PIK3CAKDM4ENPC1ALDH1A1
SCHEMBL17065998 0.77 MAP3K5 (0.53) MAP3K5ROCK2KDM4ENPC1ALDH1A1
SCHEMBL14247285 0.77 MAP3K5 (0.61) MAP3K5ROCK2KDM4ENPC1ALDH1A1
SCHEMBL31286733 0.75 MAP3K5 (0.47) MAP3K5ROCK2KDM4ESMN1; SMN2
SCHEMBL31286952 0.74 SMN1; SMN2 (0.50) MAP3K5KDM4EALDH1A1SMN1; SMN2TSHR
SCHEMBL1302695 0.74 MAP3K5 (0.46) MAP3K5PIK3CANPC1ALDH1A1POLB
SCHEMBL14318039 0.74 MAP3K5 (0.62) MAP3K5ROCK2NPC1RAB9ASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015134171-A1 HETEROARYLAMIDE INHIBITORS OF TBK1 TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2015-09-11 WO disclosed