SCHEMBL17066356

SCHEMBL17066356

Cc1ccc(C#Cc2nc(C)c(C)s2)cc1

nearest known ligand 0.46

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
GRM5 P41594 6/20 0.46
CA12 O43570 1/20 0.38
CA1 P00915 1/20 0.38
CA2 P00918 1/20 0.38
CA9 Q16790 1/20 0.38
KCNH2 Q12809 1/20 0.38
ATAD2 Q6PL18 1/20 0.37
ALDH1A1 P00352 2/20 0.36
GAA P10253 2/20 0.36
FFAR1 O14842 2/20 0.35
EGLN1 Q9GZT9 1/20 0.35
EGLN3 Q9H6Z9 1/20 0.35
CYP2A6 P11509 1/20 0.34
ACACB O00763 1/20 0.33
ADK P55263 1/20 0.33
KDM4E B2RXH2 1/20 0.33
RAB9A P51151 1/20 0.33
NOS1 P29475 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6310651 0.85 GRM5 (0.54) GRM5ALDH1A1GAAKDM4ERAB9A
SCHEMBL9445826 0.72 GRM5 (0.64) GRM5CA12CA1CA2CA9
SCHEMBL4457730 0.72 GRM5 (0.64) GRM5CA12CA1CA2CA9
SCHEMBL12599210 0.70 GRM5 (0.48) GRM5CA12CA1CA2CA9
SCHEMBL9715647 0.70 GRM5 (0.61) GRM5CA12CA1CA2CA9
SCHEMBL4138997 0.68 KDM4E (0.58) ALDH1A1GAAKDM4ERAB9A
SCHEMBL30278513 0.67 GRM5 (0.68) GRM5CA12CA1CA2CA9
SCHEMBL10060648 0.65 GRM5 (0.47) GRM5CA12CA1CA2CA9
SCHEMBL17378288 0.65 GRM5 (0.61) GRM5CA12CA1CA2CA9
SCHEMBL873622 0.65

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9127021-B2 Hepatitis C virus inhibitors ENANTA PHARMACEUTICALS, INC. (US) 2015-09-08 US disclosed