SCHEMBL17066830

SCHEMBL17066830

CC(F)(F)Cn1c(=O)n(CCO)c2nc(N)nc(NN)c21

nearest known ligand 0.32

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
PIK3CA P42336 2/20 0.32
PDE4A P27815 1/20 0.30
PDE4B Q07343 1/20 0.30
PDE4C Q08493 1/20 0.30
PDE4D Q08499 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15261253 0.90 PIK3CA (0.31) PIK3CA
SCHEMBL871896 0.84 TSHR (0.37) PIK3CAPDE4APDE4BPDE4CPDE4D
SCHEMBL872848 0.82 ADORA2A (0.36) PDE4APDE4BPDE4CPDE4D
SCHEMBL872376 0.80 ALDH1A1 (0.36) PDE4APDE4BPDE4CPDE4D
SCHEMBL872488 0.77 PDE5A (0.46) PDE4APDE4BPDE4CPDE4D
SCHEMBL876961 0.75 EEF2K (0.34) PIK3CAPDE4APDE4BPDE4CPDE4D
SCHEMBL15261850 0.74 PIK3CA (0.33) PIK3CAPDE4APDE4BPDE4CPDE4D
SCHEMBL17066867 0.70 ADORA2A (0.35) PDE4APDE4BPDE4CPDE4D
SCHEMBL872374 0.67 ADORA2A (0.40) PDE4APDE4BPDE4CPDE4D
SCHEMBL874074 0.66 TSHR (0.39) PDE4APDE4BPDE4CPDE4D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2619211-B1 FUSED TRICYCLIC COMPOUNDS AS ADENOSINE RECEPTOR ANTAGONIST ADVINUS THERAPEUTICS LTD (IN) 2015-09-09 EP disclosed