SCHEMBL17067754

SCHEMBL17067754

Cc1ccc2c(ccn2-c2cccnc2)c1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ROCK1 Q13464 1/20 0.50
CYP2A6 P11509 4/20 0.49
CYP3A4 P08684 3/20 0.49
CYP2E1 P05181 2/20 0.49
CYP19A1 P11511 2/20 0.43
MAPT P10636 3/20 0.42
RXFP1 Q9HBX9 1/20 0.42
MAOB P27338 1/20 0.42
CYP11B2 P19099 4/20 0.41
CYP11B1 P15538 3/20 0.41
TSHR P16473 1/20 0.40
NPSR1 Q6W5P4 1/20 0.40
PTK2 Q05397 1/20 0.39
KDM4C Q9H3R0 1/20 0.39
FGFR1 P11362 1/20 0.39
MDM2 Q00987 1/20 0.39
KDM4E B2RXH2 1/20 0.39
MEN1 O00255 1/20 0.39
TP53 P04637 1/20 0.39
CYP1A2 P05177 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6663687 0.88 CYP11B2 (0.49) ROCK1CYP2A6CYP3A4CYP2E1CYP19A1
SCHEMBL6656915 0.86 CYP11B1 (0.50) CYP2A6CYP3A4CYP2E1CYP19A1MAPT
SCHEMBL8736804 0.82 ROCK1 (0.54) ROCK1CYP19A1MAPTRXFP1MAOB
SCHEMBL17067770 0.82 FGFR1 (0.51) ROCK1CYP2A6MAPTRXFP1MAOB
SCHEMBL30364924 0.81 MAPT (0.48) CYP2A6CYP3A4CYP2E1CYP19A1MAPT
SCHEMBL4232123 0.81 ROCK1 (0.50) ROCK1CYP2A6CYP3A4CYP2E1CYP19A1
SCHEMBL8306084 0.81 CYP19A1 (0.53) CYP2A6CYP3A4CYP2E1CYP19A1CYP11B2
SCHEMBL2264468 0.81 MAPT (0.48) CYP2A6CYP3A4CYP2E1CYP19A1MAPT
SCHEMBL21671905 0.81 MAPT (0.51) CYP2A6CYP3A4CYP2E1CYP19A1MAPT
SCHEMBL6682744 0.80 CYP11B2 (0.50) CYP2A6CYP3A4CYP2E1CYP19A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2915804-A1 NOVEL AMINE DERIVATIVE OR SALT THEREOF Toyama Chemical Co., Ltd. (JP) 2015-09-09 EP disclosed