SCHEMBL17072192

SCHEMBL17072192

Cc1ccc(C=C[C@@H](O)C(CO)N(NC(=O)OC(C)(C)C)C(=O)OC(C)(C)C)cc1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 1/20 0.35
CYP2C9 P11712 1/20 0.35
CYP2C19 P33261 1/20 0.35
PPARA Q07869 3/20 0.34
AKT1 P31749 3/20 0.34
PPARG P37231 2/20 0.34
NPC1 O15118 2/20 0.33
RAB9A P51151 2/20 0.33
MAPT P10636 2/20 0.33
KDM4E B2RXH2 1/20 0.33
MIF P14174 1/20 0.32
HDAC8 Q9BY41 2/20 0.32
HDAC6 Q9UBN7 2/20 0.32
HDAC3 O15379 1/20 0.32
HDAC4 P56524 1/20 0.32
HDAC1 Q13547 1/20 0.32
HDAC7 Q8WUI4 1/20 0.32
HDAC2 Q92769 1/20 0.32
HDAC10 Q969S8 1/20 0.32
HDAC11 Q96DB2 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17072191 1.00 CYP3A4 (0.35) CYP3A4CYP2C9CYP2C19PPARAAKT1
SCHEMBL17072190 1.00 CYP3A4 (0.35) CYP3A4CYP2C9CYP2C19PPARAAKT1
SCHEMBL17072195 0.91 NFKB1 (0.39) PPARAAKT1PPARGNPC1RAB9A
SCHEMBL17072193 0.91 NFKB1 (0.39) PPARAAKT1PPARGNPC1RAB9A
SCHEMBL17072194 0.91 NFKB1 (0.39) PPARAAKT1PPARGNPC1RAB9A
SCHEMBL17072206 0.83 AKT1 (0.35) CYP3A4CYP2C9CYP2C19PPARAAKT1
SCHEMBL17072205 0.83 AKT1 (0.35) CYP3A4CYP2C9CYP2C19PPARAAKT1
SCHEMBL17072207 0.83 AKT1 (0.35) CYP3A4CYP2C9CYP2C19PPARAAKT1
SCHEMBL16865339 0.83 PPARA (0.37) CYP3A4CYP2C9CYP2C19PPARANPC1
SCHEMBL16859610 0.79 CYP3A4 (0.41) CYP3A4CYP2C9CYP2C19PPARANPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9133488-B2 Synthetic methods and compounds related thereto UNIVERSITY OF ALASKA FAIRBANKS (US) 2015-09-15 US disclosed