SCHEMBL17078958

SCHEMBL17078958

O=C(O)N1CCCC(Cn2ccc3cc(Br)ccc32)CC1

nearest known ligand 0.49

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
HTR7 P34969 3/20 0.44
KRAS P01116 2/20 0.42
ACHE P22303 1/20 0.42
KDM2B Q8NHM5 2/20 0.40
NTSR1 P30989 1/20 0.40
CNR1 P21554 1/20 0.40
F2 P00734 1/20 0.40
FABP3 P05413 1/20 0.39
FABP2 P12104 1/20 0.39
FABP4 P15090 1/20 0.39
FABP5 Q01469 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17063344 0.84 SMN1; SMN2 (0.47) ACHEF2
SCHEMBL17063383 0.83 KDM4E (0.46) ACHEF2
SCHEMBL17063266 0.80 POLB (0.50) ACHEF2
SCHEMBL17063253 0.79 FPR2 (0.48) KRAS
SCHEMBL1581511 0.79 KMT2A (0.53)
SCHEMBL17063326 0.79 SMN1; SMN2 (0.51) F2
SCHEMBL17063250 0.75 SMN1; SMN2 (0.47) F2
SCHEMBL17458530 0.75 CHRM1 (0.48) HTR7FABP4
SCHEMBL17063357 0.74 HTR2A (0.47) HTR7KRASNTSR1
Hydrochloric Acid SCHEMBL17063302 0.73 HTR2A (0.46) HTR7KRAS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3116504-A2 RETINOIC ACID RECEPTOR-RELATED ORPHAN RECEPTOR MODULATORS AND USES THEREOF Innov17 LLC (US) 2017-01-18 EP disclosed
WO-2015138276-A2 RETINOIC ACID RECEPTOR-RELATED ORPHAN RECEPTOR MODULATORS AND USES THEREOF INNOV17 LLC (US) 2015-09-17 WO disclosed