SCHEMBL1707953

SCHEMBL1707953

CC(C(=O)O)[C@@H]1COc2cc(N)ccc21

nearest known ligand 0.39

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
LTB4R Q15722 8/20 0.39
LTB4R2 Q9NPC1 8/20 0.39
CHRNB4 P30926 4/20 0.36
CHRNA3 P32297 4/20 0.36
CHRNB2 P17787 1/20 0.36
CHRNA4 P43681 1/20 0.36
PTGS1 P23219 1/20 0.33
PTGS2 P35354 1/20 0.33
ALDH1A1 P00352 1/20 0.33
PPARG P37231 2/20 0.32
PPARD Q03181 2/20 0.32
FFAR1 O14842 1/20 0.32
ACHE P22303 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3502661 1.00 LTB4R (0.39) LTB4RLTB4R2CHRNB4CHRNA3CHRNB2
SCHEMBL204322 0.84 LTB4R (0.40) LTB4RLTB4R2CHRNB4CHRNA3CHRNB2
SCHEMBL17431399 0.84 LTB4R (0.40) LTB4RLTB4R2CHRNB4CHRNA3CHRNB2
SCHEMBL205688 0.84 LTB4R (0.40) LTB4RLTB4R2CHRNB4CHRNA3CHRNB2
SCHEMBL205181 0.82 LTB4R (0.50) LTB4RLTB4R2PTGS1PTGS2PPARG
SCHEMBL5788067 0.75 PPARG (0.51) LTB4RLTB4R2PPARGPPARDFFAR1
SCHEMBL17431441 0.73 LTB4R (0.34) LTB4RLTB4R2PTGS1PTGS2ALDH1A1
SCHEMBL1707872 0.72 CHRNB4 (0.36) LTB4RLTB4R2CHRNB4CHRNA3CHRNB2
SCHEMBL2729054 0.72 GAA (0.36) LTB4RLTB4R2CHRNB4CHRNA3CHRNB2
SCHEMBL7179171 0.72 ESR1 (0.39) LTB4RLTB4R2CHRNB4CHRNA3CHRNB2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2440541-A1 NOVEL FUSED CYCLIC COMPOUND AND USE THEREOF Takeda Pharmaceutical Company Limited (JP) 2012-04-18 EP disclosed
WO-2010143733-A1 NOVEL FUSED CYCLIC COMPOUND AND USE THEREOF TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2010-12-16 WO disclosed