SCHEMBL17080683

SCHEMBL17080683

CC(C)c1ccc(-c2ccc3nc(C(C)(C)C)ccc3c2)cc1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 3/20 0.41
AAK1 Q2M2I8 1/20 0.38
KCNH2 Q12809 1/20 0.36
HRH3 Q9Y5N1 1/20 0.36
RAB9A P51151 4/20 0.35
MAPT P10636 3/20 0.35
PAX8 Q06710 1/20 0.35
NOD2 Q9HC29 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
DHODH Q02127 2/20 0.34
PTPN5 P54829 2/20 0.34
NPC1 O15118 3/20 0.33
SMN1; SMN2 Q16637 2/20 0.33
SCN4A P35499 1/20 0.33
HDAC6 Q9UBN7 2/20 0.33
TP53 P04637 2/20 0.33
HDAC3 O15379 1/20 0.33
HDAC1 Q13547 1/20 0.33
HDAC2 Q92769 1/20 0.33
HDAC8 Q9BY41 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10024929 0.87 PSMB5 (0.40) BACE1KCNH2HRH3RAB9AMAPT
SCHEMBL23841257 0.85 PIK3CD (0.38) RAB9AMAPTNPC1TP53KDM4E
SCHEMBL12190334 0.83 CYP1A2 (0.44) BACE1AAK1KCNH2HRH3RAB9A
SCHEMBL12173608 0.82 KIF11 (0.44) BACE1KCNH2HRH3RAB9AMAPT
SCHEMBL12436949 0.79 CYP1A2 (0.52) BACE1AAK1KDM4EPOLBCYP1A2
SCHEMBL10120019 0.79 AAK1 (0.50) BACE1AAK1RAB9AMAPTPAX8
SCHEMBL14072407 0.78 NPC1 (0.38) KCNH2HRH3RAB9AMAPTNPC1
SCHEMBL23502417 0.78 KCNH2 (0.38) BACE1KCNH2HRH3CYP1A2PSMB5
SCHEMBL14328084 0.76 BRAF (0.38) AAK1RAB9AMAPTPAX8NOD2
SCHEMBL888873 0.73 AAK1 (0.42) BACE1AAK1RAB9AMAPTPAX8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9133170-B2 Inhibitors of HCV NS5A HOFFMANN-LA ROCHE INC. (US) 2015-09-15 US disclosed