SCHEMBL17088199

SCHEMBL17088199

CCOc1ccc(-c2nn(CCO)cc2-c2ccncc2)cc1

nearest known ligand 0.66

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.66
KMT2A Q03164 1/20 0.66
SLC6A3 Q01959 2/20 0.55
BRAF P15056 4/20 0.54
PDE10A Q9Y233 2/20 0.53
BMPR1B O00238 2/20 0.53
CIT O14578 2/20 0.53
RIPK2 O43353 2/20 0.53
STK10 O94804 2/20 0.53
MAP4K4 O95819 2/20 0.53
ABL1 P00519 2/20 0.53
RAF1 P04049 2/20 0.53
ERBB3 P21860 2/20 0.53
JAK1 P23458 2/20 0.53
ACVR1B P36896 2/20 0.53
TGFBR1 P36897 2/20 0.53
CSNK1D P48730 2/20 0.53
CSNK1E P49674 2/20 0.53
MAPK10 P53779 2/20 0.53
MAP2K5 Q13163 2/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17088989 0.91 MEN1 (0.64) MEN1KMT2ASLC6A3BRAFPDE10A
SCHEMBL17088197 0.89 SLC6A3 (0.69) SLC6A3PDE10A
SCHEMBL17088195 0.89 SLC6A3 (0.69) SLC6A3PDE10A
SCHEMBL17088189 0.84 MAPK13 (0.63) BRAFPDE10ACSNK1DCSNK1E
SCHEMBL17088192 0.84 MAPK13 (0.63) BRAFPDE10ACSNK1DCSNK1E
SCHEMBL17088202 0.83 PDE10A (0.57) MEN1KMT2ASLC6A3PDE10A
SCHEMBL17088200 0.83 MEN1 (0.62) MEN1KMT2ASLC6A3BRAFPDE10A
SCHEMBL11996180 0.82 PDE10A (0.61) SLC6A3PDE10A
SCHEMBL17088198 0.81 BRAF (0.60) MEN1KMT2ASLC6A3BRAFPDE10A
SCHEMBL1759065 0.81 SLC6A3 (0.83) MEN1KMT2ASLC6A3PDE10A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9138494-B2 Radiolabeled PDE10A ligands ABBVIE INC. (US) 2015-09-22 US disclosed