SCHEMBL17089705

SCHEMBL17089705

O=C(/N=C(\Nc1cc(C(F)(F)F)n[nH]1)NC1CCOCC1)c1ccc(Cl)cc1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC4 P56524 3/20 0.41
HDAC6 Q9UBN7 2/20 0.41
TRPV1 Q8NER1 2/20 0.38
CCNA2 P20248 2/20 0.37
CDK2 P24941 2/20 0.37
CCNA1 P78396 2/20 0.37
GABRA5 P31644 2/20 0.36
HDAC1 Q13547 1/20 0.35
HDAC2 Q92769 1/20 0.35
CNR2 P34972 1/20 0.35
ACKR3 P25106 1/20 0.35
DYRK1A Q13627 1/20 0.34
RHOC P08134 1/20 0.34
RHOA P61586 1/20 0.34
PTGS2 P35354 1/20 0.34
PDE4B Q07343 1/20 0.34
TACR2 P21452 1/20 0.33
TACR1 P25103 1/20 0.33
ANO1 Q5XXA6 1/20 0.33
GSK3B P49841 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9920694 0.93 TRPV1 (0.43) HDAC4HDAC6TRPV1CCNA2CDK2
SCHEMBL9921137 0.91 CCNA2 (0.41) HDAC4HDAC6CCNA2CDK2CCNA1
SCHEMBL9921132 0.91 HDAC4 (0.40) HDAC4HDAC6TRPV1GABRA5CNR2
SCHEMBL9920882 0.89 CNR2 (0.39) HDAC4HDAC6CCNA2CDK2CCNA1
SCHEMBL9921025 0.89 HDAC6 (0.39) HDAC4HDAC6TRPV1CDK2DYRK1A
SCHEMBL9921119 0.85 MAPK1 (0.39) HDAC4HDAC6GABRA5GSK3BKCNH2
SCHEMBL9920883 0.84 ALDH1A1 (0.47) GSK3BKCNH2
SCHEMBL9920841 0.84 CCNA2 (0.41) HDAC4HDAC6TRPV1CCNA2CDK2
SCHEMBL19041506 0.84 CCNA2 (0.35) CCNA2CDK2CCNA1RHOCRHOA
SCHEMBL9920693 0.83 TRPV1 (0.42) HDAC4HDAC6TRPV1CCNA2CDK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9139532-B2 Pyrazolyl guanidine F1F0-atpase inhibitors and therapeutic uses thereof LYCERA CORPORATION (US) 2015-09-22 US disclosed