SCHEMBL17089969

SCHEMBL17089969

COC(=O)CCCc1ccc(NCCCCCNS(=O)(=O)C(C)(C)C)cc1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTPRB P23467 2/20 0.42
EPHX2 P34913 1/20 0.41
CA12 O43570 3/20 0.41
CA7 P43166 3/20 0.41
CA9 Q16790 3/20 0.41
CA14 Q9ULX7 3/20 0.41
CA2 P00918 3/20 0.39
IDO1 P14902 1/20 0.38
ALDH1A1 P00352 2/20 0.37
KDM4E B2RXH2 1/20 0.37
GAA P10253 1/20 0.37
MAPT P10636 1/20 0.37
HSD17B10 Q99714 1/20 0.37
PKM P14618 1/20 0.37
CA1 P00915 1/20 0.37
ADRB2 P07550 1/20 0.36
ADRB1 P08588 1/20 0.36
ADRB3 P13945 1/20 0.36
PTPRC P08575 1/20 0.36
PTPN2 P17706 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17089970 0.88 NR1H4 (0.47) ALDH1A1HSD17B10PKM
SCHEMBL10113485 0.86 EPHX2 (0.47) EPHX2ALDH1A1MAPTPTPRC
SCHEMBL11935068 0.84 GRIA1 (0.44) PTPRBEPHX2CA12CA7CA9
SCHEMBL11934794 0.83 HPGD (0.46) CA12CA9CA2KDM4ECA1
SCHEMBL13438596 0.83 HPGD (0.46) CA12CA9CA2KDM4ECA1
SCHEMBL13565863 0.81 EPHX1 (0.43) CA9CA2ALDH1A1MAPTCA1
SCHEMBL13564843 0.81 HPGD (0.47) CA12CA9CA2KDM4ECA1
SCHEMBL11934940 0.80 EPHX2 (0.46) PTPRBEPHX2CA2ALDH1A1KDM4E
SCHEMBL13565491 0.80 MEN1 (0.36) CA2ALDH1A1KDM4EGAAMAPT
SCHEMBL31522321 0.79 CA12 (0.53) EPHX2CA12CA7CA9CA14

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9139518-B2 Amine derivative having NPY Y5 receptor antagonistic activity SHIONOGI & CO., LTD. (JP) 2015-09-22 US disclosed