SCHEMBL17090109

SCHEMBL17090109

CC(C)(C)S(=O)(=O)Nc1ccc(NC[C@H]2CC[C@H](NS(=O)(=O)C(C)(C)C)CC2)cc1

nearest known ligand 0.39

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.39
ALDH3A1 P30838 1/20 0.39
CNR2 P34972 7/20 0.38
NPY5R Q15761 1/20 0.37
BRD4 O60885 2/20 0.37
MET P08581 1/20 0.35
PTPN11 Q06124 1/20 0.34
CRHR1 P34998 1/20 0.34
CNR1 P21554 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13565117 1.00 ALDH1A1 (0.39) ALDH1A1ALDH3A1CNR2NPY5RBRD4
SCHEMBL17090188 0.92 ALDH1A1 (0.45) ALDH1A1ALDH3A1CNR2NPY5RMET
SCHEMBL17090359 0.89 ALDH1A1 (0.39) ALDH1A1ALDH3A1CNR2NPY5R
SCHEMBL13564865 0.89 ALDH1A1 (0.39) ALDH1A1ALDH3A1CNR2NPY5R
SCHEMBL17090161 0.89 ALDH1A1 (0.36) ALDH1A1ALDH3A1CNR2NPY5RBRD4
SCHEMBL13565586 0.89 ALDH1A1 (0.36) ALDH1A1ALDH3A1CNR2NPY5RBRD4
SCHEMBL17090312 0.88 ALDH1A1 (0.39) ALDH1A1ALDH3A1CNR2NPY5RCRHR1
SCHEMBL13213210 0.88 ALDH1A1 (0.39) ALDH1A1ALDH3A1CNR2NPY5RCRHR1
SCHEMBL13564851 0.88 NPY5R (0.41) ALDH1A1ALDH3A1CNR2NPY5RCRHR1
SCHEMBL17090166 0.88 NPY5R (0.41) ALDH1A1ALDH3A1CNR2NPY5RCRHR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9139518-B2 Amine derivative having NPY Y5 receptor antagonistic activity SHIONOGI & CO., LTD. (JP) 2015-09-22 US disclosed