SCHEMBL17090189

SCHEMBL17090189

Cc1c(NC[C@H]2CC[C@H](NS(=O)(=O)C(C)C)CC2)ccc(OC2CCCC2)c1C

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE4A P27815 2/20 0.37
SMN1; SMN2 Q16637 3/20 0.36
PI4KB Q9UBF8 2/20 0.35
PTGER4 P35408 2/20 0.35
CYP19A1 P11511 2/20 0.33
ALDH1A1 P00352 2/20 0.33
MEN1 O00255 2/20 0.33
TSHR P16473 2/20 0.33
KMT2A Q03164 2/20 0.33
ALDH3A1 P30838 1/20 0.33
PTGES O14684 1/20 0.33
CYP1A2 P05177 1/20 0.33
CYP3A4 P08684 1/20 0.33
CYP2D6 P10635 1/20 0.33
MAPT P10636 1/20 0.33
ALOX15 P16050 1/20 0.33
PTGS1 P23219 1/20 0.33
CYP2C19 P33261 1/20 0.33
PTGS2 P35354 1/20 0.33
NPY5R Q15761 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13565127 1.00 PDE4A (0.37) PDE4ASMN1; SMN2PI4KBPTGER4CYP19A1
SCHEMBL17090197 0.85 PTGER4 (0.36) PDE4ASMN1; SMN2PI4KBPTGER4NPY5R
SCHEMBL13565174 0.85 PTGER4 (0.36) PDE4ASMN1; SMN2PI4KBPTGER4NPY5R
SCHEMBL13564896 0.82 PTGS1 (0.36) PI4KBPTGER4ALDH1A1ALDH3A1PTGS1
SCHEMBL17090437 0.82 PTGS1 (0.36) PI4KBPTGER4ALDH1A1ALDH3A1PTGS1
SCHEMBL10114990 0.80 POLB (0.45) SMN1; SMN2ALDH1A1KMT2ABRD4
SCHEMBL13204435 0.80 POLB (0.45) SMN1; SMN2ALDH1A1KMT2ABRD4
SCHEMBL13564914 0.80 PDE4A (0.41) PDE4API4KBALDH1A1MEN1TSHR
SCHEMBL13439249 0.79 PTGER4 (0.41) PDE4ASMN1; SMN2PTGER4CYP19A1ALDH1A1
SCHEMBL11935507 0.79 PTGER4 (0.41) PDE4ASMN1; SMN2PTGER4CYP19A1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9139518-B2 Amine derivative having NPY Y5 receptor antagonistic activity SHIONOGI & CO., LTD. (JP) 2015-09-22 US disclosed